ENANTIOSELECTIVE SYNTHESIS OF N-BOC AND N-FMOC PROTECTED DIETHYL 4-PHOSPHONO(DIFLUOROMETHYL)-L-PHENYLALANINE - AGENTS SUITABLE FOR THE SOLID-PHASE SYNTHESIS OF PEPTIDES CONTAINING NONHYDROLYZABLE ANALOGS OF O-PHOSPHOTYROSINE

被引：94

作者：

SMYTH, MS ^{[1
]}

BURKE, TR ^{[1
]}

机构：

[1] NCI,DCT,DTP,MED CHEM LAB,BETHESDA,MD 20892

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 04期

关键词：

D O I：

10.1016/S0040-4039(00)75835-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Enantioselective convergent syntheses of N-Boc and N-Fmoc protected diethyl 4-phosphono(difluoromethyl)-L-phenylalanine are reported. le analogues of O-phosphotyrosine/

引用

页码：551 / 554

页数：4

共 16 条

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BURKE, TR
SMYTH, MS
OTAKA, A
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[7] GARBAYJAUREGUIBERRY C, 1992, INT J PEPT PROT RES, V39, P523
[8] SYNTHESIS OF ENANTIOMERICALLY PURE PROTECTED BETA-ARYL ALANINES
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WYTHES, MJ
WOOD, A
[J]. TETRAHEDRON LETTERS, 1989, 30 (43) : 5941 - 5944
[9] A NEW DIRECT METHOD FOR THE SYNTHESIS OF ENANTIOMERICALLY PURE PROTECTED ALPHA-AMINO-ACIDS
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