THROMBOXANE SYNTHETASE INHIBITORS (TXSI) - DESIGN, SYNTHESIS, AND EVALUATION OF A NOVEL SERIES OF OMEGA-PYRIDYLALKENOIC ACIDS

被引：133

作者：

KATO, K

OHKAWA, S

TERAO, S

TERASHITA, Z

NISHIKAWA, K

机构：

[1] TAKEDA CHEM IND LTD,DIV CENT RES,CHEM LABS,JUSOHONMACHI 2 CHOME,YODOGAWA KU,OSAKA 532,JAPAN

[2] TAKEDA CHEM IND LTD,DIV CENT RES,BIOL LABS,YODOGAWA KU,OSAKA 532,JAPAN

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 03期

关键词：

D O I：

10.1021/jm00381a005

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：287 / 294

页数：8

共 17 条

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[5] IMINOSULFURANES .18. PREPARATION OF IMINOSULFURANES UTILIZING DIMETHYL SULFOXIDE-OXALYL CHLORIDE REAGENT
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[6] HIGHLY SELECTIVE INHIBITORS OF THROMBOXANE SYNTHETASE .1. IMIDAZOLE DERIVATIVES
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NAKAZAWA, M
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[7] INTERACTION OF POLYCYCLIC-HYDROCARBONS WITH CYTOCHROME-P-450 .3. EFFECTS OF HYDROCARBON BINDING ON THE INTERACTION OF SOME LIGANDS WITH P-4481 HEME
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[J]. JOURNAL OF BIOCHEMISTRY, 1982, 92 (01) : 77 - 88
[8] THROMBOXANES - SELECTIVE BIOSYNTHESIS AND DISTINCT BIOLOGICAL PROPERTIES
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MINKES, M
RAZ, A
[J]. SCIENCE, 1976, 193 (4248) : 163 - 165
[9] APPLICATION OF IMIDAZOLE AS A SELECTIVE INHIBITOR OF THROMBOXANE SYNTHETASE IN HUMAN PLATELETS
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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (04) : 1716 - 1720
[10] NISHIKAWA K, 1984, 9TH INT C PHARM LOND

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