A NOVEL FORM OF DEPENDENCY OF HEPATIC EXTRACTION RATIO OF OPIOIDS INVIVO UPON THE PORTAL-VEIN CONCENTRATION OF DRUG - COMPARISON OF MORPHINE, DIAMORPHINE, FENTANYL, METHADONE AND BUPRENORPHINE IN THE CHRONICALLY CANNULATED COW

被引:10
作者
BULLINGHAM, RES
MOORE, RA
SYMONDS, HW
ALLEN, MC
BALDWIN, D
MCQUAY, HJ
机构
[1] RADCLIFFE INFIRM,NUFFIELD DEPT ANAESTHET & CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
[2] ARC,INST RES ANIM DIS,NEWBURY RG16 0NN,BERKS,ENGLAND
关键词
D O I
10.1016/0024-3205(84)90369-2
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2047 / 2056
页数:10
相关论文
共 27 条
  • [1] BAGGOT JD, 1973, AM J VET RES, V34, P571
  • [2] SOME OBSERVATIONS ON METABOLITE PRODUCTION AND UTILIZATION INVIVO BY GUT AND LIVER OF ADULT DAIRY-COWS
    BAIRD, GD
    SYMONDS, HW
    ASH, R
    [J]. JOURNAL OF AGRICULTURAL SCIENCE, 1975, 85 (OCT) : 281 - 296
  • [3] THE RADIOIMMUNOASSAY OF BUPRENORPHINE
    BARTLETT, AJ
    LLOYDJONES, JG
    RANCE, MJ
    FLOCKHART, IR
    DOCKRAY, GJ
    BENNETT, MRD
    MOORE, RA
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 18 (04) : 339 - 345
  • [4] METABOLISM OF MORPHINE AND HEROIN IN MAN
    BOERNER, U
    ABBOTT, S
    ROE, RL
    [J]. DRUG METABOLISM REVIEWS, 1975, 4 (01) : 39 - 73
  • [5] BRUNK SF, 1975, CLIN PHARMACOL THER, V16, P1039
  • [6] BUPRENORPHINE KINETICS
    BULLINGHAM, RES
    MCQUAY, HJ
    MOORE, A
    BENNETT, MRD
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1980, 28 (05) : 667 - 672
  • [7] ACUTE METHADONE KINETICS IN MAN - RELATIONSHIP TO CHRONIC STUDIES
    BULLINGHAM, RES
    MCQUAY, HJ
    PORTER, EJB
    THOMAS, D
    ALLEN, MC
    MOORE, RA
    [J]. BRITISH JOURNAL OF ANAESTHESIA, 1982, 54 (12) : 1271 - 1276
  • [8] COHN GL, 1973, P SOC EXP BIOL MED, V144, P351
  • [9] PHARMACOKINETICS OF MORPHINE AND ITS SURROGATES .4. PHARMACOKINETICS OF HEROIN AND ITS DERIVED METABOLITES IN DOGS
    GARRETT, ER
    GURKAN, T
    [J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1980, 69 (10) : 1116 - 1134
  • [10] PHARMACOKINETICS OF MORPHINE AND ITS SURROGATES .3. MORPHINE AND MORPHINE 3-MONOGLUCURONIDE PHARMACOKINETICS IN THE DOG AS A FUNCTION OF DOSE
    GARRETT, ER
    JACKSON, AJ
    [J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (06) : 753 - 771