A NOVEL GABAA ANTAGONIST [H-3] SR 95531 - MICROSCOPIC ANALYSIS OF BINDING IN THE RAT-BRAIN AND ALLOSTERIC MODULATION BY SEVERAL BENZODIAZEPINE AND BARBITURATE RECEPTOR LIGANDS

被引:44
作者
MCCABE, RT
WAMSLEY, JK
YEZUITA, JP
OLSEN, RW
机构
[1] UNIV CALIF LOS ANGELES,CTR HLTH SCI,SCH MED,DEPT PHARMACOL,LOS ANGELES,CA 90024
[2] UNIV CALIF LOS ANGELES,CTR HLTH SCI,SCH MED,BRAIN RES INST,LOS ANGELES,CA 90024
[3] UNIV UTAH,SCH MED,DEPT PHARMACOL & TOXICOL,SALT LAKE CITY,UT 84132
[4] UNIV UTAH,SCH MED,DEPT PSYCHIAT,SALT LAKE CITY,UT 84132
关键词
D O I
10.1002/syn.890020208
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:163 / 173
页数:11
相关论文
共 43 条
[1]  
BOURGUIGNON JJ, 1985, PHARMACOLOGIST, V27, P518
[2]   STRYCHNINE AS A POTENT INHIBITOR OF THE BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M .
BRAIN RESEARCH BULLETIN, 1980, 5 :681-684
[3]   INTERACTION OF PITRAZEPIN WITH THE GABA BENZODIAZEPINE RECEPTOR COMPLEX AND WITH GLYCINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 118 (1-2) :115-121
[4]   AN ARYLAMINOPYRIDAZINE DERIVATIVE OF GAMMA-AMINOBUTYRIC ACID (GABA) IS A SELECTIVE AND COMPETITIVE ANTAGONIST AT THE GABAA RECEPTOR-SITE [J].
CHAMBON, JP ;
FELTZ, P ;
HEAULME, M ;
RESTLE, S ;
SCHLICHTER, R ;
BIZIERE, K ;
WERMUTH, CG .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (06) :1832-1836
[5]  
ENNA SJ, 1977, MOL PHARMACOL, V13, P442
[6]   PROPERTIES OF GAMMA-AMINOBUTYRIC ACID (GABA) RECEPTOR-BINDING IN RAT-BRAIN SYNAPTIC MEMBRANE-FRACTIONS [J].
ENNA, SJ ;
SNYDER, SH .
BRAIN RESEARCH, 1975, 100 (01) :81-97
[7]   THE BINDING OF THE GABA AGONIST [H-3]-LABELED THIP TO RAT-BRAIN SYNAPTIC-MEMBRANES [J].
FALCH, E ;
KROGSGAARDLARSEN, P .
JOURNAL OF NEUROCHEMISTRY, 1982, 38 (04) :1123-1129
[8]   GABA BINDING AND BICUCULLINE IN SPINAL-CORD AND CORTICAL MEMBRANES FROM ADULT-RAT AND FROM MOUSE NEURONS IN CELL-CULTURE [J].
FRERE, RC ;
MACDONALD, RL ;
YOUNG, AB .
BRAIN RESEARCH, 1982, 244 (01) :145-154
[9]   PITRAZEPIN, A NOVEL GABAA ANTAGONIST [J].
GAHWILER, BH ;
MAURER, R ;
WUTHRICH, HJ .
NEUROSCIENCE LETTERS, 1984, 45 (03) :311-316
[10]   EFFECT OF GABAERGIC DRUGS ON BENZODIAZEPINE BINDING-SITE SENSITIVITY IN RAT CEREBRAL-CORTEX [J].
GALLAGER, DW ;
THOMAS, JW ;
TALLMAN, JF .
BIOCHEMICAL PHARMACOLOGY, 1978, 27 (23) :2745-2749