THE EFFECTS OF BEPRIDIL, COMPARED WITH CALCIUM-CHANNEL INHIBITORS AND CALMODULIN ANTAGONISTS ON BOTH SPONTANEOUS ACTIVITY AND CONTRACTIONS INDUCED BY POTASSIUM OR PHENYLEPHRINE IN RAT PORTAL-VEIN

被引:11
作者
CAMPBELL, JK [1 ]
WINSLOW, E [1 ]
MARSHALL, RJ [1 ]
机构
[1] ORGANON LABS LTD,DEPT PHARMACOL,SCI DEV GRP,NEWHOUSE ML1 5SH,LANARK,SCOTLAND
关键词
D O I
10.1016/0014-2999(86)90604-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:187 / 196
页数:10
相关论文
共 34 条
[1]   BEPRIDIL AND CETIEDIL - VASODILATORS WHICH INHIBIT CA-2+-DEPENDENT CALMODULIN INTERACTIONS WITH ERYTHROCYTE-MEMBRANES [J].
AGRE, P ;
VIRSHUP, D ;
BENNETT, V .
JOURNAL OF CLINICAL INVESTIGATION, 1984, 74 (03) :812-820
[2]  
ALPERT JS, 1985, PHARMATHERAPEUTICA, V4, P195
[3]   CONTRACTION IN VENOUS SMOOTH-MUSCLE INDUCED BY HYPERTONICITY - CALCIUM DEPENDENCE AND MECHANICAL CHARACTERISTICS [J].
ANDERSSO.C ;
HELLSTRA.P ;
JOHANSSO.B ;
RINGBERG, A .
ACTA PHYSIOLOGICA SCANDINAVICA, 1974, 90 (02) :451-461
[4]  
ASANO M, 1982, J PHARMACOL EXP THER, V220, P191
[5]  
Bennett MR., 1972, AUTONOMIC NEUROMUSCU
[6]  
BOND M, 1984, J PHYSIOL-LONDON, V355, P677, DOI 10.1113/jphysiol.1984.sp015445
[7]   THE MECHANISM OF THE BLOCKADE BY TRIFLUOPERAZINE OF SOME ACTIONS OF PHENYLEPHRINE ON LIVER AND SMOOTH-MUSCLE [J].
COCKS, TM ;
DILGER, P ;
JENKINSON, DH .
BIOCHEMICAL PHARMACOLOGY, 1981, 30 (20) :2873-2875
[8]   UPTAKE OF BEPRIDIL INTO ISOLATED VENTRICULAR MYOCYTES - RETENTION BY ACTIN [J].
CRAMB, G ;
DOW, JW .
BIOCHEMICAL PHARMACOLOGY, 1983, 32 (02) :227-231
[9]  
DECUNEO MF, 1983, ARCH INT PHARMACOD T, V263, P28
[10]   THE CONTRIBUTION OF CALCIUM AND POTASSIUM TO THE ALPHA-ACTION OF ADRENALINE ON SMOOTH-MUSCLE CELLS OF THE PORTAL-VEIN, PULMONARY-ARTERY AND TAENIA CECI OF THE GUINEA-PIG [J].
DENHERTOG, A ;
PIELKENROOD, J ;
RAS, R ;
VANDENAKKER, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 98 (02) :223-234