TACHYKININ ANTAGONISTS HAVE POTENT LOCAL-ANESTHETIC ACTIONS

被引:69
作者
POST, C
BUTTERWORTH, JF
STRICHARTZ, GR
KARLSSON, JA
PERSSON, CGA
机构
[1] AB DRACO,DEPT RES & DEV,BOX 34,S-22100 LUND,SWEDEN
[2] ASTRA LAKEMEDEL AB,RES & DEV LABS,S-15185 SODERTALJE,SWEDEN
[3] UNIV LUND,DEPT CLIN PHARMACOL,S-22101 LUND,SWEDEN
[4] HARVARD UNIV,BRIGHAM & WOMENS HOSP,SCH MED,ANESTHESIA RES LAB,BOSTON,MA 02115
关键词
D O I
10.1016/0014-2999(85)90008-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:347 / 354
页数:8
相关论文
共 32 条
  • [1] INTRATHECAL (D-PRO2,D-TRP7,9)-SP ELICITS HYPOALGESIA AND MOTOR BLOCKADE IN THE RAT AND ANTAGONIZES NOXIOUS RESPONSES INDUCED BY SUBSTANCE-P
    AKERMAN, B
    ROSELL, S
    FOLKERS, K
    [J]. ACTA PHYSIOLOGICA SCANDINAVICA, 1982, 114 (04): : 631 - 633
  • [2] BOIVIE J, 1975, MTP INT REV SCIENC 1, V3, P303
  • [3] COURTNEY KR, 1978, ANESTHESIOLOGY, V48, P11
  • [4] A SYNTHETIC PEPTIDE AS AN ANTAGONIST OF SUBSTANCE-P
    ENGBERG, G
    SVENSSON, TH
    ROSELL, S
    FOLKERS, K
    [J]. NATURE, 1981, 293 (5829) : 222 - 223
  • [5] ERLANGER J, 1937, ELECTRICAL SIGNS NER
  • [6] DIFFERENTIAL SENSITIVITIES OF MAMMALIAN NERVE-FIBERS TO LOCAL-ANESTHETIC AGENTS
    GISSEN, AJ
    COVINO, BG
    GREGUS, J
    [J]. ANESTHESIOLOGY, 1980, 53 (06) : 467 - 474
  • [7] 3 TACHYKININS IN MAMMALIAN BRAIN
    HARMAR, AJ
    [J]. TRENDS IN NEUROSCIENCES, 1984, 7 (03) : 57 - 60
  • [8] IMMUNOHISTOCHEMICAL EVIDENCE FOR A NEUROTOXIC ACTION OF (D-PRO2,D-TRP7,9)-SUBSTANCE-P, AN ANALOG WITH SUBSTANCE-P ANTAGONISTIC ACTIVITY
    HOKFELT, T
    VINCENT, S
    HELLSTEN, L
    ROSELL, S
    FOLKERS, K
    MARKEY, K
    GOLDSTEIN, M
    CUELLO, C
    [J]. ACTA PHYSIOLOGICA SCANDINAVICA, 1981, 113 (04): : 571 - 573
  • [9] A SUBSTANCE-P ANTAGONIST, [D-PRO2, D-TRP7,9]SP, INHIBITS INFLAMMATORY RESPONSES IN THE RABBIT EYE
    HOLMDAHL, G
    HAKANSON, R
    LEANDER, S
    ROSELL, S
    FOLKERS, K
    SUNDLER, F
    [J]. SCIENCE, 1981, 214 (4524) : 1029 - 1031
  • [10] LOCAL-ANESTHETICS SELECTIVELY INHIBIT NON-CHOLINERGIC NEURAL CONTRACTIONS IN GUINEA-PIG AIRWAYS
    KARLSSON, JA
    PERSSON, CGA
    [J]. ACTA PHYSIOLOGICA SCANDINAVICA, 1984, 120 (03): : 469 - 471