PHOTOAFFINITY-LABELING OF THE PORCINE BRAIN ALPHA-2-ADRENERGIC RECEPTOR USING A RADIOIODINATED ARYLAZIDE DERIVATIVE OF RAUWOLSCINE - IDENTIFICATION OF THE HORMONE-BINDING SUBUNIT

被引:16
作者
LANIER, SM
GRAHAM, RM
HESS, HJ
GRODSKI, A
REPASKE, MG
NUNNARI, JM
LIMBIRD, LE
HOMCY, CJ
机构
[1] HARVARD UNIV,MASSACHUSETTS GEN HOSP,SCH MED,CARDIAC UNIT,BOSTON,MA 02114
[2] PFIZER CENT RES,GROTON,CT 06380
[3] VANDERBILT UNIV,DEPT PHARMACOL,NASHVILLE,TN 37232
关键词
D O I
10.1073/pnas.83.24.9358
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:9358 / 9362
页数:5
相关论文
共 31 条
[1]   CHARACTERIZATION OF ALPHA-1-ADRENERGIC AND ALPHA-2-ADRENERGIC RECEPTORS [J].
BYLUND, DB ;
UPRICHARD, DC .
INTERNATIONAL REVIEW OF NEUROBIOLOGY, 1983, 24 :343-431
[2]  
CERIONE RA, 1986, J BIOL CHEM, V261, P3901
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]   [H-3]-LABELED RAUWOLSCINE AND [H-3]-LABELED YOHIMBINE BINDING TO RAT CEREBRAL AND HUMAN-PLATELET MEMBRANES - POSSIBLE HETEROGENEITY OF ALPHA-2-ADRENOCEPTORS [J].
CHEUNG, YD ;
BARNETT, DB ;
NAHORSKI, SR .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 84 (1-2) :79-85
[5]   4-AZIDOANILINE, A VERSATILE PROTEIN AND PEPTIDE MODIFYING AGENT FOR PHOTO AFFINITY LABELING [J].
ESCHER, EHF ;
ROBERT, H ;
GUILLEMETTE, G .
HELVETICA CHIMICA ACTA, 1979, 62 (04) :1217-1222
[6]  
GRAHAM RM, 1986, HEART CARDIOVASCULAR, V2, P1059
[7]  
GRAHAM RM, 1982, HYPERTENSION, V4, pS183
[8]   MOLECULAR CHARACTERIZATION OF ADRENERGIC-RECEPTORS [J].
HOMCY, CJ ;
GRAHAM, RM .
CIRCULATION RESEARCH, 1985, 56 (05) :635-650
[9]   PURIFICATION AND BIOCHEMICAL-CHARACTERIZATION OF ALPHA-2-ADRENERGIC RECEPTOR FROM THE RAT ADRENOCORTICAL CARCINOMA [J].
JAISWAL, RK ;
SHARMA, RK .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 130 (01) :58-64
[10]  
KAWAHARA RS, 1985, J PHARMACOL EXP THER, V233, P603