A SIMPLE PREPARATION OF CHLOROMETHYL ESTERS OF THE BLOCKED AMINO-ACIDS

被引：20

作者：

HARADA, N ^{[1
]}

HONGU, M ^{[1
]}

TANAKA, T ^{[1
]}

KAWAGUCHI, T ^{[1
]}

HASHIYAMA, T ^{[1
]}

TSUJIHARA, K ^{[1
]}

机构：

[1] TANABE SEIYAKU CO LTD,ORGAN CHEM RES LAB,2-2-50 KAWAGISHI,TODA,SAITAMA 335,JAPAN

来源：

SYNTHETIC COMMUNICATIONS | 1994年 / 24卷 / 06期

关键词：

D O I：

10.1080/00397919408011298

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthesis of various chloromethyl esters of the blocked amino acids, very useful reagents for prodrug, are described.

引用

页码：767 / 772

页数：6

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