IRREVERSIBLE ENZYME INHIBITORS .77. INHIBITORS OF THYMIDINE PHOSPHORYLASE .3. HYDROPHOBIC BONDING BY 1-SUBSTITUTED URACILS CONTAINING ADDITIONAL SUBSTITUENTS AT 5 AND 6 POSITIONS

被引：39

作者：

BAKER, BR

KAWAZU, M

SANTI, DV

SCHWAN, TJ

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1967年 / 10卷 / 03期

关键词：

D O I：

10.1021/jm00315a003

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

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页码：304 / &

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[1] NONCLASSICAL ANTIMETABOLITES .18. SIMULATION OF 5'-PHOSPHORIBOSYL BINDING .2. OMEGA-URACIL ALKANOIC ACIDS RELATED TO 2'-DEOXYURIDYLATE
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[2] IRREVERSIBLE ENZYME INHIBITORS .75. INHIBITORS OF THYMIDINE PHOSPHORTLASE .I. MODE OF RIBOFURANOSE BINDING
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[3] NONCLASSICAL ANTIMETABOLITES .26. INHIBITORS OF THYMIDINE KINASE .2. INHIBITION BY FUNCTIONALIZED 1-ALKYLURACILS
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[4] IRREVERSIBLE ENZYME INHIBITORS .80. INHIBITORS OF THYMIDINE PHOSPHORYLASE .6. HYDROPHOBIC BONDING WITH 6 SUBSTITUENTS ON ACIDIC 5-NITRO- AND 5-BROMOURACILS
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[5] ANALOGS OF TETRAHYDROFOLIC ACID .24. FACILE SYNTHETIC ROUTE TO 2-AMINO-5-(3-ANILINOPROPYL)-6-METHYL-4-PYRIMIDINOL TYPE OF FOLIC REDUCTASE + THYMIDYLATE SYNTHETASE INHIBITOR
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[6] IRREVERSIBLE ENZYME INHIBITORS .76. INHIBITORS OF THYMIDINE PHOSPHORYLASE .2. HYDROPHOBIC BONDING BY 1-SUBSTITUTED URACILS
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (03) : 302 - &
[7] IRREVERSIBLE ENZYME INHIBITORS .78. INHIBITORS OF THYMIDINE PHOSPHORYLASE .4. HYDROPHOBIC BONDING BY URACILS SUBSTITUTED AT 5 AND 6 POSITIONS
BAKER, BR
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (03) : 311 - &
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[J]. JOURNAL OF ORGANIC CHEMISTRY, 1960, 25 (10) : 1731 - 1734
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