5-HT3 RECEPTORS MEDIATE INHIBITION OF ACETYLCHOLINE-RELEASE IN CORTICAL TISSUE

被引:237
作者
BARNES, JM [1 ]
BARNES, NM [1 ]
COSTALL, B [1 ]
NAYLOR, RJ [1 ]
TYERS, MB [1 ]
机构
[1] GLAXO GRP RES LTD,DEPT NEUROPHARMACOL,WARE SG12 ODP,HERTS,ENGLAND
关键词
D O I
10.1038/338762a0
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:762 / 763
页数:2
相关论文
共 20 条
  • [1] BARNES JM, IN PRESS BRAIN RES
  • [2] [H-3] ZACOPRIDE - LIGAND FOR THE IDENTIFICATION OF 5-HT3 RECOGNITION SITES
    BARNES, NM
    COSTALL, B
    NAYLOR, RJ
    [J]. JOURNAL OF PHARMACY AND PHARMACOLOGY, 1988, 40 (08) : 548 - 551
  • [3] PHARMACOLOGICAL PROPERTIES OF GR38032F, A NOVEL ANTAGONIST AT 5-HT3 RECEPTORS
    BUTLER, A
    HILL, JM
    IRELAND, SJ
    JORDAN, CC
    TYERS, MB
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1988, 94 (02) : 397 - 412
  • [4] EFFECTS OF THE 5-HT3 RECEPTOR ANTAGONIST, GR38032F, ON RAISED DOPAMINERGIC ACTIVITY IN THE MESOLIMBIC SYSTEM OF THE RAT AND MARMOSET BRAIN
    COSTALL, B
    DOMENEY, AM
    NAYLOR, RJ
    TYERS, MB
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1987, 92 (04) : 881 - 894
  • [5] ZACOPRIDE - ANXIOLYTIC PROFILE IN RODENT AND PRIMATE MODELS OF ANXIETY
    COSTALL, B
    DOMENEY, AM
    GERRARD, PA
    KELLY, ME
    NAYLOR, RJ
    [J]. JOURNAL OF PHARMACY AND PHARMACOLOGY, 1988, 40 (04) : 302 - 305
  • [6] EFFECT OF QUIPAZINE, A SEROTONIN-LIKE DRUG, ON STRIATAL CHOLINERGIC INTERNEURONES
    EUVRARD, C
    JAVOY, F
    HERBERT, A
    GLOWINSKI, J
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 41 (03) : 281 - 289
  • [7] BLOCKADE OF NEURONAL TRYPTAMINE RECEPTORS BY METOCLOPRAMIDE
    FOZARD, JR
    MOBAROKALI, ATM
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 49 (01) : 109 - 112
  • [8] SEROTONIN INHIBITS ACETYLCHOLINE-RELEASE FROM RAT STRIATUM SLICES - EVIDENCE FOR A PRESYNAPTIC RECEPTOR-MEDIATED EFFECT
    GILLET, G
    AMMOR, S
    FILLION, G
    [J]. JOURNAL OF NEUROCHEMISTRY, 1985, 45 (06) : 1687 - 1691
  • [9] EFFECT OF THE 5-HT3 RECEPTOR ANTAGONIST, GR38032F, ON RESPONSES TO INJECTION OF A NEUROKININ AGONIST INTO THE VENTRAL TEGMENTAL AREA OF THE RAT-BRAIN
    HAGAN, RM
    BUTLER, A
    HILL, JM
    JORDAN, CC
    IRELAND, SJ
    TYERS, MB
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 138 (02) : 303 - 305
  • [10] HOYER DT, 1988, PHARM SCI, V9, P89