INHIBITION OF SERINE PROTEASES BY PEPTIDYL FLUOROMETHYL KETONES

被引：268

作者：

IMPERIALI, B ^{[1
]}

ABELES, RH ^{[1
]}

机构：

[1] BRANDEIS UNIV,GRAD DEPT BIOCHEM,WALTHAM,MA 02254

来源：

BIOCHEMISTRY | 1986年 / 25卷 / 13期

关键词：

D O I：

10.1021/bi00361a005

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：3760 / 3767

页数：8

共 34 条

[1] THE SLOW, TIGHT-BINDING INHIBITION OF CATHEPSIN-B BY LEUPEPTIN - A HYSTERETIC EFFECT [J].

BAICI, A ;

GYGERMARAZZI, M .

EUROPEAN JOURNAL OF BIOCHEMISTRY, 1982, 129 (01) :33-41

[2] PHOSPHONAMIDATES AS TRANSITION-STATE ANALOG INHIBITORS OF THERMOLYSIN [J].

BARTLETT, PA ;

MARLOWE, CK .

BIOCHEMISTRY, 1983, 22 (20) :4618-4624

[3] ELASTASE-CATALYZED HYDROLYSIS OF P-NITROPHENYL TRIMETHYLACETATE [J].

BENDER, ML ;

MARSHALL, TH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1968, 90 (01) :201-&

[4] CRYSTALLOGRAPHIC AND KINETIC INVESTIGATIONS OF THE COVALENT COMPLEX FORMED BY A SPECIFIC TETRAPEPTIDE ALDEHYDE AND THE SERINE PROTEASE FROM STREPTOMYCES-GRISEUS [J].

BRAYER, GD ;

DELBAERE, LTJ ;

JAMES, MNG ;

BAUER, CA ;

THOMPSON, RC .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (01) :96-100

[5] BINDING OF SPECIFIC AND NONSPECIFIC ALDEHYDE SUBSTRATE ANALOGS TO ALPHA-CHYMOTRYPSIN [J].

BREAUX, EJ ;

BENDER, ML .

FEBS LETTERS, 1975, 56 (01) :81-84

[6] SENSITIVE SUBSTRATES FOR HUMAN-LEUKOCYTE AND PORCINE PANCREATIC ELASTASE - STUDY OF THE MERITS OF VARIOUS CHROMOPHORIC AND FLUOROGENIC LEAVING GROUPS IN ASSAYS FOR SERINE PROTEASES [J].

CASTILLO, MJ ;

NAKAJIMA, K ;

ZIMMERMAN, M ;

POWERS, JC .

ANALYTICAL BIOCHEMISTRY, 1979, 99 (01) :53-64

[7] TIGHT-BINDING INHIBITORS .1. KINETIC-BEHAVIOR [J].

CHA, S .

BIOCHEMICAL PHARMACOLOGY, 1975, 24 (23) :2177-2185

[8] EVIDENCE FOR HEMIACETAL FORMATION BETWEEN N-ACYL-L-PHENYLALANINALS AND ALPHA-CHYMOTRYPSIN BY CROSS-SATURATION NUCLEAR MAGNETIC-RESONANCE SPECTROSCOPY [J].

CHEN, R ;

GORENSTEIN, DG ;

KENNEDY, WP ;

LOWE, G ;

NURSE, D ;

SCHULTZ, RM .

BIOCHEMISTRY, 1979, 18 (05) :921-926

[9] FLUORO KETONE INHIBITORS OF HYDROLYTIC ENZYMES [J].

GELB, MH ;

SVAREN, JP ;

ABELES, RH .

BIOCHEMISTRY, 1985, 24 (08) :1813-1817

[10] CARBONYL ADDITION-REACTIONS - FACTORS AFFECTING HYDRATE-HEMIACETAL AND HEMIACETAL-ACETAL EQUILIBRIUM-CONSTANTS [J].

GUTHRIE, JP .

CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE, 1975, 53 (06) :898-906

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