THE PREPARATION AND LITHIATION OF BROMOFLUOROFURANS VIA A NOVEL FLUORODECARBOXYLATION

被引：19

作者：

FORREST, AK

OHANLON, PJ

机构：

[1] SmithKline Beecham Pharmaceuticals, Betchworth, Surrey RH3 7AJ, Brockham Park

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 12期

关键词：

D O I：

10.1016/0040-4039(95)00170-H

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The fluorodecarboxylation of bromofuroic acids using Selectfluor(TM) reagent 1 gives bromofluorofurans which can be lithiated and reacted with electrophiles to yield 3- or 5-substituted 2-fluorofurans.

引用

页码：2117 / 2118

页数：2

共 11 条

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