PHOSPHOLIPID-SENSITIVE CA-2+-DEPENDENT PROTEIN-KINASE INHIBITION BY R-24571, A CALMODULIN ANTAGONIST

被引：69

作者：

MAZZEI, GJ

SCHATZMAN, RC

TURNER, RS

VOGLER, WR

KUO, JF

机构：

[1] EMORY UNIV,SCH MED,DEPT PHARMACOL,ATLANTA,GA 30322

[2] EMORY UNIV,SCH MED,DEPT MED,DIV HEMATOL & ONCOL,ATLANTA,GA 30322

来源：

BIOCHEMICAL PHARMACOLOGY | 1984年 / 33卷 / 01期

关键词：

D O I：

10.1016/0006-2952(84)90379-4

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：125 / 130

页数：6

共 30 条

[1] THE ANTI-CALMODULIN DRUGS TRIFLUOPERAZINE AND R24571 REMOVE THE ACTIVATION OF THE PURIFIED ERYTHROCYTE CA-2+-ATPASE BY ACIDIC PHOSPHOLIPIDS AND BY CONTROLLED PROTEOLYSIS [J].

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FEBS LETTERS, 1982, 143 (01) :65-68

[2]

BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3

[3] R-24571 - A NEW POWERFUL INHIBITOR OF RED-BLOOD-CELL CA++-TRANSPORT ATPASE AND OF CALMODULIN-REGULATED FUNCTIONS [J].

GIETZEN, K ;

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BADER, H .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1981, 101 (02) :418-425

[4]

HELFMAN DM, 1983, CANCER RES, V43, P2955

[5]

HIDAKA H, 1979, BIOCHEM BIOPH RES CO, V90, P649

[6]

HO HC, 1977, J BIOL CHEM, V252, P43

[7]

KANAMORI M, 1981, J PHARMACOL EXP THER, V217, P494

[8] INHIBITION BY MELITTIN OF PHOSPHOLIPID-SENSITIVE AND CALMODULIN-SENSITIVE CA-2+-DEPENDENT PROTEIN-KINASES [J].

KATOH, N ;

RAYNOR, RL ;

WISE, BC ;

SCHATZMAN, RC ;

TURNER, RS ;

HELFMAN, DM ;

FAIN, JN ;

KUO, JF .

BIOCHEMICAL JOURNAL, 1982, 202 (01) :217-224

[9] DIFFERENTIAL REGULATION OF CALCIUM DEPENDENT AND CALCIUM INDEPENDENT CYCLIC-NUCLEOTIDE PHOSPHODIESTERASES FROM HEART BY PALMITOYLCARNITINE AND PALMITOYL COENZYME-A [J].

KATOH, N ;

HELFMAN, DM ;

WRENN, RW ;

KUO, JF .

BIOCHIMICA ET BIOPHYSICA ACTA, 1982, 714 (01) :129-135

[10] COBRA POLYPEPTIDE CYTOTOXIN-I AND MARINE WORM POLYPEPTIDE CYTOTOXIN-A-IV ARE POTENT AND SELECTIVE INHIBITORS OF PHOSPHOLIPID-SENSITIVE CA-2+-DEPENDENT PROTEIN-KINASE [J].

KUO, JF ;

RAYNOR, RL ;

MAZZEI, GJ ;

SCHATZMAN, RC ;

TURNER, RS ;

KEM, WR .

FEBS LETTERS, 1983, 153 (01) :183-186

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