INTERACTIONS OF QUINIDINE AND QUININE AND (+)-PINDOLOL AND (-)-PINDOLOL WITH THE ORGANIC CATION PROTON ANTIPORTER IN RENAL BRUSH-BORDER MEMBRANE-VESICLES

被引:20
作者
OTT, RJ
HUI, AC
WONG, FM
HSYU, PH
GIACOMINI, KM
机构
[1] UNIV CALIF SAN FRANCISCO,MED CTR,SCH PHARM,BOX 0446,SAN FRANCISCO,CA 94143
[2] UNIV CALIF SAN FRANCISCO,MED CTR,SCH MED,SAN FRANCISCO,CA 94143
关键词
D O I
10.1016/0006-2952(91)90023-X
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:142 / 145
页数:4
相关论文
共 30 条
[1]   CHIRALITY IN BIOACTIVE AGENTS AND ITS PITFALLS [J].
ARIENS, EJ .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1986, 7 (05) :200-205
[2]  
Booth A G, 1974, Biochem J, V142, P575
[3]   CIMETIDINE TRANSPORT IN ISOLATED LUMINAL MEMBRANE-VESICLES FROM RABBIT KIDNEY [J].
GISCLON, L ;
WONG, FM ;
GIACOMINI, KM .
AMERICAN JOURNAL OF PHYSIOLOGY, 1987, 253 (01) :F141-F150
[4]   QUANTITATIVE RELATIONSHIPS BETWEEN STRUCTURE AND PHARMACOKINETICS OF BETA-ADRENOCEPTOR BLOCKING-AGENTS IN MAN [J].
HINDERLING, PH ;
SCHMIDLIN, O ;
SEYDEL, JK .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1984, 12 (03) :263-287
[5]  
HNSCH C, 1979, SUBSTITUENT CONSTANT, P13
[6]  
HOLOHAN PD, 1981, J PHARMACOL EXP THER, V216, P294
[7]  
HSYU PH, 1988, DRUG METAB DISPOS, V16, P503
[8]   INTERACTIONS OF ORGANIC-ANIONS WITH THE ORGANIC CATION TRANSPORTER IN RENAL BBMV [J].
HSYU, PH ;
GISCLON, LG ;
HUI, AC ;
GIACOMINI, KM .
AMERICAN JOURNAL OF PHYSIOLOGY, 1988, 254 (01) :F56-F61
[9]   ESSENTIAL TYROSINE RESIDUES IN TRANSPORT OF ORGANIC CATIONS IN RENAL BBMV [J].
HSYU, PH ;
GIACOMINI, KM .
AMERICAN JOURNAL OF PHYSIOLOGY, 1987, 252 (06) :F1065-F1072
[10]   STEREOSELECTIVE RENAL CLEARANCE OF PINDOLOL IN HUMANS [J].
HSYU, PH ;
GIACOMINI, KM .
JOURNAL OF CLINICAL INVESTIGATION, 1985, 76 (05) :1720-1726