5,9-METHANOBENZOANNULENAMINES .1. IMPROVED SYNTHESIS OF 11-AMINO-5,9-METHANOBENZO[8]ANNULENES

被引：4

作者：

GILBERT, IM ^{[1
]}

HEWETT, CL ^{[1
]}

RAE, DR ^{[1
]}

REDPATH, J ^{[1
]}

SAVAGE, DS ^{[1
]}

SLEIGH, T ^{[1
]}

机构：

[1] ORGANON RES LABS LTD,ORGANON SCI DEV GRP,MOTHERWELL ML1 5SH,SCOTLAND

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1995年 / 02期

关键词：

D O I：

10.1039/p19950000133

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Reaction of 1-(3,4-dihydronapthalen-2-yl) pyrrolidine with acrylaldehyde gave an epimeric mixture of 8-hydroxy-5,6,7,8,9,10-hexahydro-5,9-methanobenzo[8]annulen-11-ones which was used for the synthesis of several 11-amino derivatives.

引用

页码：133 / 139

页数：7

共 15 条

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