NEW EFFECTIVE GONADOTROPIN-RELEASING-HORMONE ANTAGONISTS WITH MINIMAL POTENCY FOR HISTAMINE-RELEASE INVITRO

被引：153

作者：

RIVIER, JE ^{[1
]}

PORTER, J ^{[1
]}

RIVIER, CL ^{[1
]}

PERRIN, M ^{[1
]}

CORRIGAN, A ^{[1
]}

HOOK, WA ^{[1
]}

SIRAGANIAN, RP ^{[1
]}

VALE, WW ^{[1
]}

机构：

[1] NIDR,MICROBIOL & IMMUNOL LAB,CLIN IMMUNOL SECT,BETHESDA,MD 20892

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 10期

关键词：

D O I：

10.1021/jm00160a008

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1846 / 1851

页数：6

共 29 条

[1]

CORBIN A, 1975, ENDOCR RES COMMUN, V2, P1

[2]

Coy DH, 1981, LHRH PEPTIDES FEMALE, P37

[3]

DITTMER K, 1948, J BIOL CHEM, V173, P323

[4]

DUTTA AS, 1985, ANNU REP MED CHEM, V20, P203

[5] MODIFICATION OF PEPTIDES CONTAINING GLUTAMIC-ACID BY HYDROGEN FLUORIDE-ANISOLE MIXTURES - GAMMA-ACYLATION OF ANISOLE OR GLUTAMYL NITROGEN [J].

FEINBERG, RS ;

MERRIFIELD, RB .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1975, 97 (12) :3485-3496

[6] ANTAGONISTS OF THE LUTEINIZING-HORMONE RELEASING HORMONE WITH PYRIDYL-ALANINES WHICH COMPLETELY INHIBIT OVULATION AT NANOGRAM DOSAGE [J].

FOLKERS, K ;

BOWERS, CY ;

KUBIAK, T ;

STEPINSKI, J .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 111 (03) :1089-1095

[7]

HOES C, 1980, RECL TRAV CHIM PAY B, V99, P99

[8]

HOOK WA, 1985, FED PROC, V44, P1323

[9] GONADOTROPIN-RELEASING-HORMONE ANALOG DESIGN - STRUCTURE-FUNCTION STUDIES TOWARD THE DEVELOPMENT OF AGONISTS AND ANTAGONISTS - RATIONALE AND PERSPECTIVE [J].

KARTEN, MJ ;

RIVIER, JE .

ENDOCRINE REVIEWS, 1986, 7 (01) :44-66

[10]

KARTEN MJ, LHRH ITS ANALOGS, V2

← 1 2 3 →