3'-ISOPROPYL-3,5-DIIODO-L-THYRONINE - A POTENT SYNTHETIC THYROMIMETIC THYRONINE ANALOG - STUDIES OF ITS KINETICS AND BIOLOGICAL POTENCY IN MAN AND RATS AND ITS TOXICOLOGY

被引:9
作者
KAISER, CA [1 ]
SALOMONMONTAVON, NA [1 ]
MERKELBACH, U [1 ]
BURGER, AG [1 ]
机构
[1] UNIV GENEVA, DEPT MED, DIV ENDOCRINOL, THYROID RES UNIT, CH-1211 GENEVA 4, SWITZERLAND
关键词
D O I
10.1210/jcem-57-1-44
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:44 / 49
页数:6
相关论文
共 12 条
[1]  
BURGER AG, 1980, 6TH INT C END MELB, P479
[2]   RELATIVE ACTIVITIES OF SERVERAL 3'-AND 3'-5'- ALKYL AND ARYL THYROMIMETIC AGENTS [J].
GREENBERG, CM ;
BLANK, B ;
PAULS, JF ;
PFEIFFER, FR .
AMERICAN JOURNAL OF PHYSIOLOGY, 1963, 205 (05) :821-&
[3]  
KOERNER D, 1975, J BIOL CHEM, V250, P6417
[4]  
NETER J, 1974, APPLIED LINEAR STATI
[5]   LIMITED BINDING-CAPACITY SITES FOR L-TRIIODOTHYRONINE IN RAT-LIVER NUCLEI - NUCLEAR-CYTOPLASMIC INTERRELATION, BINDING CONSTANTS, AND CROSS-REACTIVITY WITH L-THYROXINE [J].
OPPENHEIMER, JH ;
SCHWARTZ, HL ;
KOERNER, D ;
SURKS, MI .
JOURNAL OF CLINICAL INVESTIGATION, 1974, 53 (03) :768-777
[6]   CORRECTION [J].
OPPENHEIMER, JH .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1975, 41 (06) :1172-1173
[7]   DETERMINATION OF COMMON PARAMETERS OF IODOTHYRONINE METABOLISM AND DISTRIBUTION IN MAN BY NONCOMPARTMENTAL ANALYSIS [J].
OPPENHEIMER, JH ;
SCHWARTZ, HL ;
SURKS, MI .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1975, 41 (02) :319-324
[8]   EFFECT OF THYROID-HORMONE ANALOGS ON DISPLACEMENT OF I-125-L-TRIIODOTHYRO-9 FROM HEPATIC AND HEART NUCLEI IN-VIVO - POSSIBLE RELATIONSHIP TO HORMONAL ACTIVITY [J].
OPPENHEIMER, JH ;
SCHWARTZ, HL ;
DILLMAN, W ;
SURKS, MI .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1973, 55 (03) :544-550
[9]  
PITTMAN CS, 1974, HDB PHYSIOL, V3, P233
[10]  
SILVA ES, 1977, J BIOL CHEM, V252, P6799