CALCIUM-CHANNEL AGONIST AND ANTAGONIST EFFECTS OF THE STEREOISOMERS OF THE DIHYDROPYRIDINE 202-791

被引:59
作者
KONGSAMUT, S [1 ]
KAMP, TJ [1 ]
MILLER, RJ [1 ]
SANGUINETTI, MC [1 ]
机构
[1] GD SEARLE & CO,DEPT BIOL,SKOKIE,IL 60201
关键词
D O I
10.1016/0006-291X(85)90393-6
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:141 / 148
页数:8
相关论文
共 11 条
[1]   CALCIUM-CHANNEL ACTIVATION - A DIFFERENT TYPE OF DRUG-ACTION [J].
FREEDMAN, SB ;
MILLER, RJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (17) :5580-5583
[2]  
FREEDMAN SB, 1984, J NEUROSCI, V4, P1453
[3]   DIFFERENT MODES OF CA-CHANNEL GATING BEHAVIOR FAVORED BY DIHYDROPYRIDINE CA-AGONISTS AND ANTAGONISTS [J].
HESS, P ;
LANSMAN, JB ;
TSIEN, RW .
NATURE, 1984, 311 (5986) :538-544
[4]  
HOF RP, 1985, J CARDIOVASC PHARM
[5]  
KAMP TJ, 1985, BRIT J PHARM
[6]   INTERACTION OF STEROIDAL ALKALOID TOXINS WITH CALCIUM CHANNELS IN NEURONAL CELL-LINES [J].
KONGSAMUT, S ;
FREEDMAN, SB ;
SIMON, BE ;
MILLER, RJ .
LIFE SCIENCES, 1985, 36 (15) :1493-1501
[7]   HOW MANY TYPES OF CALCIUM CHANNELS EXIST IN NEURONS [J].
MILLER, RJ .
TRENDS IN NEUROSCIENCES, 1985, 8 (02) :45-47
[8]   REGULATION OF CARDIAC CALCIUM-CHANNEL CURRENT AND CONTRACTILE ACTIVITY BY THE DIHYDROPYRIDINE BAY K-8644 IS VOLTAGE-DEPENDENT [J].
SANGUINETTI, MC ;
KASS, RS .
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 1984, 16 (07) :667-670
[9]   THE EFFECTS OF DIHYDROPYRIDINES ON NEUROTRANSMITTER RELEASE FROM CULTURED NEURONAL CELLS [J].
SHALABY, IA ;
KONGSAMUT, S ;
FREEDMAN, SB ;
MILLER, RJ .
LIFE SCIENCES, 1984, 35 (12) :1289-1295
[10]  
THOMAS G, 1985, J CARDIOVASC PHARM