DIAZEPAM ENHANCES THE ACTION BUT NOT THE BINDING OF THE GABA ANALOG, THIP

被引:13
作者
SKERRITT, JH [1 ]
MACDONALD, RL [1 ]
机构
[1] UNIV MICHIGAN,MED CTR,DEPT NEUROL,ANN ARBOR,MI 48109
关键词
D O I
10.1016/0006-8993(84)90557-2
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:181 / 186
页数:6
相关论文
共 26 条
[1]   PHARMACOLOGICAL EVIDENCE FOR 2 KINDS OF GABA RECEPTOR ON RAT HIPPOCAMPAL PYRAMIDAL CELLS STUDIED INVITRO [J].
ALGER, BE ;
NICOLL, RA .
JOURNAL OF PHYSIOLOGY-LONDON, 1982, 328 (JUL) :125-141
[2]   GAMMA-AMINOBUTYRIC ACID AGONISTS - AN INVITRO COMPARISON BETWEEN DEPRESSION OF SPINAL SYNAPTIC ACTIVITY AND DEPOLARIZATION OF SPINAL ROOT FIBERS IN THE RAT [J].
ALLAN, RD ;
EVANS, RH ;
JOHNSTON, GAR .
BRITISH JOURNAL OF PHARMACOLOGY, 1980, 70 (04) :609-615
[3]  
BARKER JL, 1981, AMINO ACID NEUROTRAN, P281
[4]   PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M ;
KROGSGAARDLARSEN, P ;
FALCH, E .
NATURE, 1979, 280 (5720) :331-333
[5]   BENZODIAZEPINES IN TREATMENT OF EPILEPSY - REVIEW [J].
BROWNE, TR ;
PENRY, JK .
EPILEPSIA, 1973, 14 (03) :277-310
[6]   CHLORDIAZEPOXIDE SELECTIVELY AUGMENTS GABA ACTION IN SPINAL-CORD CELL-CULTURES [J].
CHOI, DW ;
FARB, DH ;
FISCHBACH, GD .
NATURE, 1977, 269 (5626) :342-344
[7]   THE BINDING OF THE GABA AGONIST [H-3]-LABELED THIP TO RAT-BRAIN SYNAPTIC-MEMBRANES [J].
FALCH, E ;
KROGSGAARDLARSEN, P .
JOURNAL OF NEUROCHEMISTRY, 1982, 38 (04) :1123-1129
[8]   ENDOGENOUS PROTEIN MODULATES AFFINITY OF GABA AND BENZODIAZEPINE RECEPTORS IN RAT-BRAIN [J].
GUIDOTTI, A ;
TOFFANO, G ;
COSTA, E .
NATURE, 1978, 275 (5680) :553-555
[9]  
HAEFELY W, 1981, HDB EXPT PHARM 2, V55, P13
[10]   ANALGESIC PROPERTIES OF THE GABA-MINETIC THIP [J].
HILL, RC ;
MAURER, R ;
BUESCHER, HH ;
ROEMER, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 69 (02) :221-224