NA+ CHANNELS AS SITES OF ACTION OF THE CARDIOACTIVE AGENT DPI 201-106 WITH AGONIST AND ANTAGONIST ENANTIOMERS

被引:67
作者
ROMEY, G
QUAST, U
PAURON, D
FRELIN, C
RENAUD, JF
LAZDUNSKI, M
机构
[1] CNRS,CTR BIOCHIM,F-06034 NICE,FRANCE
[2] LABS SANDOZ,DIV PHARMACEUT,RECH PRECLIN,CH-4002 BASEL,SWITZERLAND
关键词
D O I
10.1073/pnas.84.3.896
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:896 / 900
页数:5
相关论文
共 30 条
[1]   EFFECTS OF NEUROTOXINS (VERATRIDINE, SEA-ANEMONE TOXIN, TETRODOTOXIN) ON TRANSMITTER ACCUMULATION AND RELEASE BY NERVE-TERMINALS INVITRO [J].
ABITA, JP ;
CHICHEPORTICHE, R ;
SCHWEITZ, H ;
LAZDUNSKI, M .
BIOCHEMISTRY, 1977, 16 (09) :1838-1844
[2]  
BARHANIN J, 1982, J BIOL CHEM, V257, P2553
[3]   SIMPLIFIED REAL-TIME TELEVISION IMAGE ANALYZER BASED ON AN APPLE-II MICROCOMPUTER [J].
BORDES, M ;
BERNENGO, JC ;
RENAUD, JF .
REVIEW OF SCIENTIFIC INSTRUMENTS, 1983, 54 (08) :1053-1058
[4]  
BRODY TM, 1984, PHARM CARDIAC GLYCOS, P405
[5]   THE ROLE OF SODIUM-CHANNELS IN THE EFFECTS OF THE CARDIOTONIC COMPOUND DPI 201-106 ON CONTRACTILITY AND MEMBRANE-POTENTIALS IN ISOLATED MAMMALIAN HEART PREPARATIONS [J].
BUGGISCH, D ;
ISENBERG, G ;
RAVENS, U ;
SCHOLTYSIK, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 118 (03) :303-311
[7]  
CATTERALL WA, 1981, J BIOL CHEM, V256, P8922
[8]   SYNTHESIS OF NEW, HIGHLY RADIOACTIVE TETRODOTOXIN DERIVATIVES AND THEIR BINDING-PROPERTIES TO THE SODIUM-CHANNEL [J].
CHICHEPORTICHE, R ;
BALERNA, M ;
LOMBET, A ;
ROMEY, G ;
LAZDUNSKI, M .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1980, 104 (02) :617-625
[9]  
CREVELING CR, 1983, MOL PHARMACOL, V23, P350
[10]   THE OPTICAL ISOMERS OF THE 1,4-DIHYDROPYRIDINE BAY K-8644 SHOW OPPOSITE EFFECTS ON CA CHANNELS [J].
FRANCKOWIAK, G ;
BECHEM, M ;
SCHRAMM, M ;
THOMAS, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 114 (02) :223-226