LOSS OF PIRENZEPINE REGIONAL SELECTIVITY FOLLOWING SOLUBILIZATION AND PARTIAL-PURIFICATION OF THE PUTATIVE M1 AND M2 MUSCARINIC RECEPTOR SUBTYPES

被引:8
作者
BAUMGOLD, J [1 ]
MERRIL, C [1 ]
GERSHON, ES [1 ]
机构
[1] NIMH,CLIN NEUROGENET BRANCH,BETHESDA,MD 20892
来源
MOLECULAR BRAIN RESEARCH | 1987年 / 2卷 / 01期
关键词
D O I
10.1016/0169-328X(87)90015-5
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:7 / 14
页数:8
相关论文
共 23 条
[1]   PURIFICATION OF MUSCARINIC ACETYLCHOLINE-RECEPTORS BY AFFINITY-CHROMATOGRAPHY [J].
ANDRE, C ;
DEBACKER, JP ;
GUILLET, JC ;
VANDERHEYDEN, P ;
VAUQUELIN, G ;
STROSBERG, AD .
EMBO JOURNAL, 1983, 2 (04) :499-504
[2]   OLIGOMERIC STRUCTURE OF MUSCARINIC RECEPTORS IS SHOWN BY PHOTOAFFINITY-LABELING - SUBUNIT ASSEMBLY MAY EXPLAIN HIGH-AFFINITY AND LOW-AFFINITY AGONIST STATES [J].
AVISSAR, S ;
AMITAI, G ;
SOKOLOVSKY, M .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (01) :156-159
[3]  
BIRDSALL NJM, 1978, MOL PHARMACOL, V14, P723
[4]   THE BINDING OF PIRENZEPINE TO DIGITONIN-SOLUBILIZED MUSCARINIC ACETYLCHOLINE-RECEPTORS FROM THE RAT MYOCARDIUM [J].
BIRDSALL, NJM ;
HULME, EC ;
KEEN, M .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 87 (02) :307-316
[5]  
BROWN JH, 1985, MOL PHARMACOL, V27, P525
[6]   MUSCARINIC CHOLINERGIC RECEPTOR OF RAT-BRAIN - FACTORS INFLUENCING MIGRATION IN ELECTROPHORESIS AND GEL-FILTRATION IN SODIUM DODECYL-SULFATE [J].
DADI, HK ;
MORRIS, RJ .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1984, 144 (03) :617-628
[7]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[8]   RECEPTOR-STIMULATED INOSITOL PHOSPHOLIPID-METABOLISM IN THE CENTRAL NERVOUS-SYSTEM [J].
DOWNES, CP .
CELL CALCIUM, 1982, 3 (4-5) :413-428
[9]  
FISHER SK, 1983, J BIOL CHEM, V258, P7358
[10]  
HAGA K, 1985, J BIOL CHEM, V260, P7927