SELECTIVE-INHIBITION OF STEROIDOGENIC P450 ENZYMES - CURRENT STATUS AND FUTURE PERSPECTIVES

被引：27

作者：

HARTMANN, RW

机构：

[1] Fachrichtung 12.1 Pharmazeutische Chemie, Universität des Saarlandes, D-66041 Saarbrücken

来源：

EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | 1994年 / 2卷 / 1-2期

关键词：

D O I：

10.1016/0928-0987(94)90052-3

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

[No abstract available]

引用

页码：15 / 16

页数：2

共 8 条

[1] NEW AROMATASE INHIBITORS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF PYRIDYL-SUBSTITUTED TETRALONE DERIVATIVES [J].

BAYER, H ;

BATZL, C ;

HARTMANN, RW ;

MANNSCHRECK, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (09) :2685-2691

[2] FADROZOLE HYDROCHLORIDE - A POTENT, SELECTIVE, NONSTEROIDAL INHIBITOR OF AROMATASE FOR THE TREATMENT OF ESTROGEN-DEPENDENT DISEASE [J].

BROWNE, LJ ;

GUDE, C ;

RODRIGUEZ, H ;

STEELE, RE ;

BHATNAGER, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (02) :725-736

[3] MECHANISM AND INHIBITION OF CYTOCHROME-P-450 AROMATASE [J].

COLE, PA ;

ROBINSON, CH .

JOURNAL OF MEDICINAL CHEMISTRY, 1990, 33 (11) :2933-2942

[4] NEW NONSTEROIDAL AROMATASE INHIBITORS - FOCUS ON R76713 [J].

DECOSTER, R ;

WOUTERS, W ;

BOWDEN, CR ;

VANDEN BOSSCHE, H ;

BRUYNSEELS, J ;

TUMAN, RW ;

VANGINCKEL, R ;

SNOECK, E ;

VANPEER, A ;

JANSSEN, PAJ .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1990, 37 (03) :335-341

[5] SYNTHESIS AND AROMATASE INHIBITION OF 3-CYCLOALKYL-SUBSTITUTED 3-(4-AMINOPHENYL)PIPERIDINE-2,6-DIONES [J].

HARTMANN, RW ;

BATZL, C ;

PONGRATZ, TM ;

MANNSCHRECK, A .

JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (12) :2210-2214

[6]

HARTMANN RW, 1994, 207TH ACS NAT M SAN

[7]

SERGEJEW T, 1994, IN PRESS J ENZ INHIB

[8] IS THERE A CASE FOR P-450 INHIBITORS IN CANCER-TREATMENT [J].

VANWAUWE, JP ;

JANSSEN, PAJ .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (10) :2231-2239

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