A 3-STATE MODEL OF THE BENZODIAZEPINE RECEPTOR EXPLAINS THE INTERACTIONS BETWEEN THE BENZODIAZEPINE ANTAGONIST RO 15-1788, BENZODIAZEPINE TRANQUILIZERS, BETA-CARBOLINES, AND PHENOBARBITONE

被引:318
作者
POLC, P
BONETTI, EP
SCHAFFNER, R
HAEFELY, W
机构
关键词
D O I
10.1007/BF00498510
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:260 / 264
页数:5
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共 34 条
[1]  
AHLQUIST J, 1982, BRIT J PHARMACOL, V75, pP48
[2]   HIPPOCAMPAL SEIZURES AND FAILURE OF INHIBITION [J].
BENARI, Y ;
KRNJEVIC, K ;
REINHARDT, W .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1979, 57 (12) :1462-1466
[3]   ACTION OF PICROTOXIN ON PRESYNAPTIC INHIBITION OF VARIOUS ORIGINS IN CATS SPINAL CORD [J].
BESSON, JM ;
RIVOT, JP ;
ALEONARD, P .
BRAIN RESEARCH, 1971, 26 (01) :212-&
[4]   BENZODIAZEPINE ANTAGONIST RO 15-1788 - NEUROLOGICAL AND BEHAVIORAL-EFFECTS [J].
BONETTI, EP ;
PIERI, L ;
CUMIN, R ;
SCHAFFNER, R ;
PIERI, M ;
GAMZU, ER ;
MULLER, RKM ;
HAEFELY, W .
PSYCHOPHARMACOLOGY, 1982, 78 (01) :8-18
[5]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[6]   URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M ;
OLSEN, CE .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2288-2292
[7]   PROCONVULSANT EFFECTS IN BABOONS OF BETA-CARBOLINE, A PUTATIVE ENDOGENOUS LIGAND FOR BENZODIAZEPINE RECEPTORS [J].
CEPEDA, C ;
TANAKA, T ;
BESSELIEVRE, R ;
POTIER, P ;
NAQUET, R ;
ROSSIER, J .
NEUROSCIENCE LETTERS, 1981, 24 (01) :53-57
[8]   CHLORDIAZEPOXIDE SELECTIVELY POTENTIATES GABA CONDUCTANCE OF SPINAL-CORD AND SENSORY NEURONS IN CELL-CULTURE [J].
CHOI, DW ;
FARB, DH ;
FISCHBACH, GD .
JOURNAL OF NEUROPHYSIOLOGY, 1981, 45 (04) :621-631
[9]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[10]  
COURVOISIER SIMONE, 1956, JOUR CLIN AND EXPTL PSYCHOPATH AND QUART REV PSYCHIATRY AND NEUROL, V17, P25