NEW APPLICATION OF AMINO-ACID N-CARBOXY ANHYDRIDES - SYNTHESIS OF 1,4-BENZODIAZEPINE-2,5-DIONES

被引：7

作者：

AKSSIRA, M

KASMI, H

DAHDOUH, A

BOUMZEBRA, M

机构：

[1] Université Abdelmalek Essaadi, Fac des Sciences Laboratoire de Chimie Organique B.P.2121, Tétouan

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 14期

关键词：

D O I：

10.1016/S0040-4039(00)74168-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A new synthetic method for 1,4-benzodiazepine-2,5-dione (BZD) was accomplished by the coupling of amino acid N-carboxy anhydrides (NCAs) with Bocanthranilic acid, followed by the deprotection of Boc group and by the ring expansion.

引用

页码：1887 / 1888

页数：2

共 10 条

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