N-2-(2,4-DINITROPHENYL)ETHYLOXYCARBONYL-AMINO ACIDS, NEW BASE LABILE PROTECTED DERIVATIVES SUITABLE FOR SOLID-PHASE PEPTIDE-SYNTHESIS

被引：7

作者：

ACEDO, M

ALBERICIO, F

ERITJA, R

机构：

[1] CSIC,CID,DEPT MOLEC GENET,JORDI GIRONA 18-26,E-08034 BARCELONA,SPAIN

[2] UNIV BARCELONA,DEPT ORGAN CHEM,E-08028 BARCELONA,SPAIN

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 34期

关键词：

AMINO PROTECTION; SOLID PHASE PEPTIDE SYNTHESIS; 9-FLUORENYLMETHYLOXYCARBONYL; BETA-ELIMINATION;

D O I：

10.1016/S0040-4039(00)61253-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The base labile N-2-(2,4-dinitrophenyl)ethyloxycarbonyl (Dnpeoc) group has been developed for the protection of the alpha-amino group of amino acids. Preparation of DnPeoc-amino acids and their application to solid-phase peptide synthesis are described.

引用

页码：4989 / 4992

页数：4

共 12 条

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[5]

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[6]

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