BREMAZOCINE IS AN AGONIST AT KAPPA-OPIOID RECEPTORS AND AN ANTAGONIST AT MU-OPIOID RECEPTORS IN THE GUINEA-PIG MYENTERIC PLEXUS

被引：60

作者：

CORBETT, AD

KOSTERLITZ, HW

机构：

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 1986年 / 89卷 / 01期

关键词：

D O I：

10.1111/j.1476-5381.1986.tb11141.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

收藏

页码：245 / 249

页数：5

相关论文

共 17 条

[1] SOME QUANTITATIVE USES OF DRUG ANTAGONISTS
ARUNLAKSHANA, O
SCHILD, HO
[J]. BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01): : 48 - 58
[2] SPECIFIC RECEPTOR FOR THE OPIOID PEPTIDE DYNORPHIN - STRUCTURE-ACTIVITY-RELATIONSHIPS
CHAVKIN, C
GOLDSTEIN, A
[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (10): : 6543 - 6547
[3] CORBETT A D, 1985, British Journal of Pharmacology, V86, p704P
[4] SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR
CORBETT, AD
GILLAN, MGC
KOSTERLITZ, HW
MCKNIGHT, AT
PATERSON, SJ
ROBSON, LE
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (01) : 271 - 279
[5] PRE-INCUBATION OF GUINEA-PIG MYENTERIC PLEXUS WITH BETA-FUNALTREXAMINE - DISCREPANCY BETWEEN BINDING ASSAYS AND BIOASSAYS
CORBETT, AD
KOSTERLITZ, HW
MCKNIGHT, AT
PATERSON, SJ
ROBSON, LE
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1985, 85 (03) : 665 - 673
[6] UNEXPECTED ANTAGONISM IN THE RAT VAS-DEFERENS BY BENZOMORPHANS WHICH ARE AGONISTS IN OTHER PHARMACOLOGICAL TESTS
GILLAN, MGC
KOSTERLITZ, HW
MAGNAN, J
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1981, 72 (01) : 13 - 15
[7] GOLDSTEIN A, 1984, MOL PHARMACOL, V25, P343
[8] ASSESSMENT IN GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN DEPENDENT MONKEY
HUTCHINSON, M
KOSTERLITZ, HW
LESLIE, FM
WATERFIELD, AA
TERENIUS, L
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1975, 55 (04) : 541 - 546
[9] KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS WITH PARTICULAR REFERENCE TO N-ALLYLNOROXYMORPHONE (NALOXONE)
KOSTERLITZ, HW
WATT, AJ
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (02) : 266 - +
[10] THE BINDING SPECTRUM OF NARCOTIC ANALGESIC DRUGS WITH DIFFERENT AGONIST AND ANTAGONIST PROPERTIES
MAGNAN, J
PATERSON, SJ
TAVANI, A
KOSTERLITZ, HW
[J]. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 319 (03) : 197 - 205