ANTAGONISTS WITH NEGATIVE INTRINSIC ACTIVITY AT DELTA-OPIOID RECEPTORS COUPLED TO GTP-BINDING PROTEINS

被引:458
作者
COSTA, T [1 ]
HERZ, A [1 ]
机构
[1] MAX PLANCK INST PSYCHIAT, DEPT NEUROPHARMACOL, D-8033 MARTINSRIED, GERMANY
关键词
D O I
10.1073/pnas.86.19.7321
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:7321 / 7325
页数:5
相关论文
共 39 条
[1]  
AKTORIES K, 1982, MOL PHARMACOL, V21, P336
[2]   SODIUM-IONS INCREASE THE BINDING OF THE ANTAGONIST PEPTIDE ICI-174864 TO THE DELTA-OPIATE RECEPTOR [J].
APPELMANS, N ;
CARROLL, JA ;
RANCE, MJ ;
SIMON, EJ ;
TRAYNOR, JR .
NEUROPEPTIDES, 1986, 7 (02) :139-143
[3]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[4]  
ASANO T, 1986, MOL PHARMACOL, V29, P244
[5]   RECONSTITUTION OF CATECHOLAMINE-STIMULATED BINDING OF GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE) TO THE STIMULATORY GTP-BINDING PROTEIN OF ADENYLATE-CYCLASE [J].
ASANO, T ;
PEDERSEN, SE ;
SCOTT, CW ;
ROSS, EM .
BIOCHEMISTRY, 1984, 23 (23) :5460-5467
[6]   INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
SCHMIECHEN, R ;
NEEF, G ;
NIELSEN, M ;
PETERSEN, EN .
SCIENCE, 1982, 216 (4551) :1241-1243
[7]   RECIPROCAL MODULATION OF AGONIST AND ANTAGONIST BINDING TO MUSCARINIC CHOLINERGIC RECEPTOR BY GUANINE-NUCLEOTIDE [J].
BURGISSER, E ;
DELEAN, A ;
LEFKOWITZ, RJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (06) :1732-1736
[8]   CATECHOLAMINE-STIMULATED GTPASE ACTIVITY IN TURKEY ERYTHROCYTE-MEMBRANES [J].
CASSEL, D ;
SELINGER, Z .
BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 452 (02) :538-551
[9]   THE MAMMALIAN BETA-2-ADRENERGIC RECEPTOR - RECONSTITUTION OF FUNCTIONAL INTERACTIONS BETWEEN PURE RECEPTOR AND PURE STIMULATORY NUCLEOTIDE BINDING-PROTEIN OF THE ADENYLATE-CYCLASE SYSTEM [J].
CERIONE, RA ;
CODINA, J ;
BENOVIC, JL ;
LEFKOWITZ, RJ ;
BIRNBAUMER, L ;
CARON, MG .
BIOCHEMISTRY, 1984, 23 (20) :4519-4525
[10]   OPIOID-PEPTIDES INDUCE REDUCTION OF ENKEPHALIN RECEPTORS IN CULTURED NEURO-BLASTOMA CELLS [J].
CHANG, KJ ;
ECKEL, RW ;
BLANCHARD, SG .
NATURE, 1982, 296 (5856) :446-448