PHARMACOKINETIC EVALUATION OF UK-49,858, A METABOLICALLY STABLE TRIAZOLE ANTIFUNGAL DRUG, IN ANIMALS AND HUMANS

被引:310
作者
HUMPHREY, MJ [1 ]
JEVONS, S [1 ]
TARBIT, MH [1 ]
机构
[1] PFIZER LTD,CENT RES,SANDWICH,KENT,ENGLAND
关键词
D O I
10.1128/AAC.28.5.648
中图分类号
Q93 [微生物学];
学科分类号
071005 ; 100705 ;
摘要
引用
收藏
页码:648 / 653
页数:6
相关论文
共 18 条
  • [1] KETOCONAZOLE, AN ORAL ANTIFUNGAL - LABORATORY AND CLINICAL-ASSESSMENT OF IMIDAZOLE DRUGS
    BORELLI, D
    FUENTES, J
    LEIDERMAN, E
    RESTREPO, A
    BRAN, JL
    LEGENDRE, R
    LEVINE, HB
    STEVENS, DA
    [J]. POSTGRADUATE MEDICAL JOURNAL, 1979, 55 (647) : 657 - 661
  • [2] DISPOSITION OF KETOCONAZOLE, AN ORAL ANTIFUNGAL, IN HUMANS
    BRASS, C
    GALGIANI, JN
    BLASCHKE, TF
    DEFELICE, R
    OREILLY, RA
    STEVENS, DA
    [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1982, 21 (01) : 151 - 158
  • [3] SYSTEMIC ANTIFUNGAL POTENTIAL, SAFETY, BIOTRANSPORT AND TRANSFORMATION OF MICONAZOLE NITRATE
    BRUGMANS, J
    VANCUTSE.J
    HEYKANTS, J
    SCHUERMANS, V
    THIENPONT, D
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1972, 5 (02) : 93 - 99
  • [4] CLINICAL PHARMACOKINETICS OF SYSTEMIC ANTI-FUNGAL DRUGS
    DANESHMEND, TK
    WARNOCK, DW
    [J]. CLINICAL PHARMACOKINETICS, 1983, 8 (01) : 17 - 42
  • [5] PHARMACOKINETICS OF KETOCONAZOLE IN NORMAL SUBJECTS
    DANESHMEND, TK
    WARNOCK, DW
    TURNER, A
    ROBERTS, CJC
    [J]. JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1981, 8 (04) : 299 - 304
  • [6] TREATMENT OF FUNGAL MENINGITIS WITH MICONAZOLE
    DERESINSKI, SC
    LILLY, RB
    LEVINE, HB
    GALGIANI, JN
    STEVENS, DA
    [J]. ARCHIVES OF INTERNAL MEDICINE, 1977, 137 (09) : 1180 - 1185
  • [7] DUHM B, 1974, POSTGRAD MED J, V50, P13
  • [8] THERAPEUTIC FAILURES WITH MICONAZOLE
    FISHER, JF
    DUMA, RJ
    MARKOWITZ, SM
    SHADOMY, S
    ESPINELINGROFF, A
    CHEW, WH
    [J]. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1978, 13 (06) : 965 - 968
  • [9] Gascoigne E.R., 1981, CLIN RES REV, V1, P177
  • [10] GIBALDI M, 1982, PHARMACOKINETICS