INHIBITION OF CATHEPSIN-D BY SUBSTRATE-ANALOGS CONTAINING STATINE AND BY ANALOGS OF PEPSTATIN

被引：35

作者：

AGARWAL, NS ^{[1
]}

RICH, DH ^{[1
]}

机构：

[1] UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 12期

关键词：

D O I：

10.1021/jm00162a015

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2519 / 2524

页数：6

共 36 条

[1] AN IMPROVED CATHEPSIN-D SUBSTRATE AND ASSAY PROCEDURE
AGARWAL, N
RICH, DH
[J]. ANALYTICAL BIOCHEMISTRY, 1983, 130 (01) : 158 - 165
[2] [Anonymous], 1972, J BIOL CHEM, V247, P977
[3] Barrett A, 1977, PROTEINASES MAMMALIA, P209
[4] NOVEL RENIN INHIBITORS CONTAINING THE AMINO-ACID STATINE
BOGER, J
LOHR, NS
ULM, EH
POE, M
BLAINE, EH
FANELLI, GM
LIN, TY
PAYNE, LS
SCHORN, TW
LAMONT, BI
VASSIL, TC
STABILITO, II
VEBER, DF
RICH, DH
BOPARI, AS
[J]. NATURE, 1983, 303 (5912) : 81 - 84
[5] RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE
BOGER, J
PAYNE, LS
PERLOW, DS
LOHR, NS
POE, M
BLAINE, EH
ULM, EH
SCHORN, TW
LAMONT, BI
LIN, TY
KAWAI, M
RICH, DH
VEBER, DF
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) : 1779 - 1790
[6] BOGER J, 1983, PEPTIDES STRUCTURE F, P569
[7] 3-DIMENSIONAL STRUCTURE OF THE COMPLEX OF THE RHIZOPUS-CHINENSIS CARBOXYL PROTEINASE AND PEPSTATIN AT 2.5-A RESOLUTION
BOTT, R
SUBRAMANIAN, E
DAVIES, DR
[J]. BIOCHEMISTRY, 1982, 21 (26) : 6956 - 6962
[8] TIGHT-BINDING INHIBITORS .2. NON-STEADY STATE NATURE OF INHIBITION OF MILK XANTHINE-OXIDASE BY ALLOPURINOL AND ALLOXANTHINE AND OF HUMAN ERYTHROCYTIC ADENOSINE DEAMINASE BY COFORMYCIN
CHA, S
AGARWAL, RP
PARKS, RE
[J]. BIOCHEMICAL PHARMACOLOGY, 1975, 24 (23) : 2187 - 2197
[9] IMMUNOINHIBITION OF INTRACELLULAR PROTEIN DIGESTION IN MACROPHAGES
DINGLE, JT
POOLE, AR
LAZARUS, GS
BARRETT, AJ
[J]. JOURNAL OF EXPERIMENTAL MEDICINE, 1973, 137 (05) : 1124 - 1141
[10] EVIN G, 1983, PEPTIDES STRUCTURE F, P583

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