A UNIQUELY POTENT RENIN INHIBITOR AND ITS UNANTICIPATED PLASMA-BINDING COMPONENT

被引：15

作者：

EVANS, BE ^{[1
]}

RITTLE, KE ^{[1
]}

BOCK, MG ^{[1
]}

BENNETT, CD ^{[1
]}

DIPARDO, RM ^{[1
]}

BOGER, J ^{[1
]}

POE, M ^{[1
]}

ULM, EH ^{[1
]}

LAMONT, BI ^{[1
]}

BLAINE, EH ^{[1
]}

FANELLI, GM ^{[1
]}

STABILITO, II ^{[1
]}

VEBER, DF ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 12期

关键词：

D O I：

10.1021/jm00150a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1755 / 1756

页数：2

共 17 条

[1] DIPEPTIDE ANALOGS - SYNTHESIS OF A POTENT RENIN INHIBITOR
BOCK, MG
DIPARDO, RM
EVANS, BE
RITTLE, KE
BOGER, JS
FREIDINGER, RM
VEBER, DF
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1985, (03) : 109 - 110
[2] NOVEL RENIN INHIBITORS CONTAINING THE AMINO-ACID STATINE
BOGER, J
LOHR, NS
ULM, EH
POE, M
BLAINE, EH
FANELLI, GM
LIN, TY
PAYNE, LS
SCHORN, TW
LAMONT, BI
VASSIL, TC
STABILITO, II
VEBER, DF
RICH, DH
BOPARI, AS
[J]. NATURE, 1983, 303 (5912) : 81 - 84
[3] BOGER J, 1983, PEPTIDES STRUCTURE F, P569
[4] COMPETITIVE INHIBITORS OF RENIN INHIBITORS EFFECTIVE AT PHYSIOLOGICAL PH
BURTON, J
POULSEN, K
HABER, E
[J]. BIOCHEMISTRY, 1975, 14 (17) : 3892 - 3898
[5] A SUBSTRATE-ANALOG INHIBITOR OF RENIN THAT IS EFFECTIVE INVIVO
CODY, RJ
BURTON, J
EVIN, G
POULSEN, K
HERD, JA
HABER, E
[J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 97 (01) : 230 - 235
[6] SOLUBLE PEPSTATINS - NEW APPROACH TO BLOCKADE INVIVO OF THE RENIN-ANGIOTENSIN SYSTEM
EVIN, G
GARDES, J
KREFT, C
CASTRO, B
CORVOL, P
MENARD, J
[J]. CLINICAL SCIENCE AND MOLECULAR MEDICINE, 1978, 55 : S167 - S169
[7] POE M, 1984, J BIOL CHEM, V259, P8358
[8] COMPETITIVE INHIBITORS OF RENIN
POULSEN, K
BURTON, J
HABER, E
[J]. BIOCHEMISTRY, 1973, 12 (20) : 3877 - 3882
[9] SPECIFICITY OF HUMAN RENIN - STUDIES WITH PEPTIDE INHIBITORS
POULSEN, K
HABER, E
BURTON, J
[J]. BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 452 (02) : 533 - 537
[10] SYNTHESIS OF ANALOGS OF THE CARBOXYL PROTEASE INHIBITOR PEPSTATIN - EFFECT OF STRUCTURE ON INHIBITION OF PEPSIN AND RENIN
RICH, DH
SUN, ETO
ULM, E
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (01) : 27 - 33

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