FUNCTIONAL-GROUP METABOLISM OF DOPAMINE-2 AGONISTS - CONVERSION OF 4-(2-DI-NORMAL-PROPYLAMINOETHYL)-2-(3H)-INDOLONE TO 4-(2-DI-NORMAL-PROPYLAMINOETHYL)-7-HYDROXY-2-(3H)-INDOLONE

被引：18

作者：

MICO, BA

SWAGZDIS, JE

FEDEROWICZ, DA

STRAUB, K

机构：

来源：

JOURNAL OF PHARMACEUTICAL SCIENCES | 1986年 / 75卷 / 10期

关键词：

D O I：

10.1002/jps.2600751003

中图分类号：

R914 [药物化学];

学科分类号：

100701 [药物化学];

摘要：

引用

页码：929 / 933

页数：5

共 22 条

[1]

DOMESTICATION OF CHEMISTRY BY DESIGN OF SAFER CHEMICALS - STRUCTURE-ACTIVITY-RELATIONSHIPS [J].

ARIENS, EJ .

DRUG METABOLISM REVIEWS, 1984, 15 (03) :425-504

[2]

NONCOMPARTMENTAL DETERMINATION OF THE STEADY-STATE VOLUME OF DISTRIBUTION [J].

BENET, LZ ;

GALEAZZI, RL .

JOURNAL OF PHARMACEUTICAL SCIENCES, 1979, 68 (08) :1071-1074

[3]

4-[2-(DI-NORMAL-PROPYLAMINO)ETHYL]-2(3H)-INDOLONE - A PREJUNCTIONAL DOPAMINE RECEPTOR AGONIST [J].

GALLAGHER, G ;

LAVANCHY, PG ;

WILSON, JW ;

HIEBLE, JP ;

DEMARINIS, RM .

JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (10) :1533-1536

[4]

DECREASED RATE OF METABOLISM INDUCED BY A SHIFT OF DOUBLE-BOND IN PROSTAGLANDIN F-2ALPHA FROM DELTA-5 TO DELTA-4 POSITION [J].

GREEN, K ;

SAMUELSSON, B ;

MAGERLEIN, BJ .

EUROPEAN JOURNAL OF BIOCHEMISTRY, 1976, 62 (03) :527-537

[5]

METABOLISM OF 2 PGF2-ALPHA ANALOGS IN PRIMATES - 15(S)-15-METHYL-DELTA-4-CIS-PGF1-ALPHA AND 16,16-DIMETHYL-DELTA-4-CIS-PGF1-ALPHA [J].

HANSSON, G .

PROSTAGLANDINS, 1979, 18 (05) :745-771

[6]

HIEBLE P, 1985, FED P FED AM SOC EXP, V44, P1465

[7]

QUANTITATIVE RELATIONSHIPS BETWEEN STRUCTURE AND PHARMACOKINETICS OF BETA-ADRENOCEPTOR BLOCKING-AGENTS IN MAN [J].

HINDERLING, PH ;

SCHMIDLIN, O ;

SEYDEL, JK .

JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1984, 12 (03) :263-287

[8]

4-(AMINOALKYL)-7-HYDROXY-2(3H)-INDOLONES, A NOVEL CLASS OF POTENT PRE-SYNAPTIC DOPAMINE RECEPTOR AGONISTS [J].

HUFFMAN, WF ;

HALL, RF ;

GRANT, JA ;

WILSON, JW ;

HIEBLE, JP ;

HAHN, RA .

JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (07) :933-935

[9]

JAKOBY WB, 1980, METABOLIC BASIS DETO, V2, P1

[10]

SYNTHESIS AND BIOLOGICAL PROPERTIES OF 16-ALKYLPROSTAGLANDINS [J].

MAGERLEI.BJ ;

DUCHARME, DW ;

MAGEE, WE ;

MILLER, WL ;

ROBERT, A ;

WEEKS, JR .

PROSTAGLANDINS, 1973, 4 (01) :143-145

← 1 2 3 →