AN IMPROVED SYNTHESIS OF 2'-DEOXY-5-AZACYTIDINE BY CONDENSATION OF A 9-FLUORENYLMETHOXYCARBONYL-PROTECTED SUGAR ONTO THE SILYLATED BASE

被引：11

作者：

BENHATTAR, J ^{[1
]}

JIRICNY, J ^{[1
]}

机构：

[1] FRIEDRICH MIESCHER INST,CH-4002 BASEL,SWITZERLAND

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1986年 / 51卷 / 16期

关键词：

D O I：

10.1021/jo00366a028

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：3211 / 3213

页数：3

共 20 条

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[3] SIDE REACTIONS IN PEPTIDE-SYNTHESIS .11. POSSIBLE REMOVAL OF THE 9-FLUORENYLMETHYLOXYCARBONYL GROUP BY THE AMINO COMPONENTS DURING COUPLING
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[5] THE FLUOREN-9-YLMETHOXYCARBONYL GROUP FOR THE PROTECTION OF HYDROXY-GROUPS - ITS APPLICATION IN THE SYNTHESIS OF AN OCTATHYMIDYLIC ACID FRAGMENT
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[6] GREEN TW, 1981, PROTECTIVE GROUPS OR, P225
[7] THE 9-FLUORENYLMETHOXYCARBONYL (FMOC) GROUP FOR THE PROTECTION OF AMINO FUNCTIONS OF CYTIDINE, ADENOSINE, GUANOSINE AND THEIR 2'-DEOXYSUGAR DERIVATIVES
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[8] ALPHA-THYMIDIN
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[9] EFFECTS OF 5-AZACYTIDINE AND ITS 2'-DEOXYDERIVATIVE ON CELL-DIFFERENTIATION AND DNA METHYLATION
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[J]. PHARMACOLOGY & THERAPEUTICS, 1985, 28 (01) : 17 - 27
[10] HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC ANALYSIS OF CHEMICAL-STABILITY OF 5-AZA-2'-DEOXYCYTIDINE
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[J]. JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (11) : 1228 - 1232

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