THE DESIGN AND SYNTHESIS OF THE ANGIOTENSIN CONVERTING-ENZYME-INHIBITOR CILAZAPRIL AND RELATED BICYCLIC COMPOUNDS

被引：90

作者：

ATTWOOD, MR ^{[1
]}

HASSALL, CH ^{[1
]}

KROHN, A ^{[1
]}

LAWTON, G ^{[1
]}

REDSHAW, S ^{[1
]}

机构：

[1] ROCHE PROD LTD,WELWYN GARDEN CIT AL7 3AY,HERTS,ENGLAND

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1986年 / 06期

关键词：

D O I：

10.1039/p19860001011

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1011 / 1019

页数：9

共 26 条

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NIXON, JS
REDSHAW, S
THOMAS, WA
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[3] BECKER R H A, 1983, Naunyn-Schmiedeberg's Archives of Pharmacology, V324, pR42
[4] INHIBITION OF ANGIOTENSIN-CONVERTING ENZYME BY ANALOGS OF PEPTIDES FROM BOTHROPS-JARARACA VENOM
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[6] GAVRAS H, 1981, LANCET, V2, P543
[7] ANTIHYPERTENSIVE EFFECT OF ORAL ANGIOTENSIN CONVERTING-ENZYME INHIBITOR SQ 14225 IN MAN
GAVRAS, H
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[10] THE DESIGN AND SYNTHESIS OF NEW TRIAZOLO, PYRAZOLO-PYRIDAZINE, AND PYRIDAZO-PYRIDAZINE DERIVATIVES AS INHIBITORS OF ANGIOTENSIN CONVERTING ENZYME
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MOODY, CJ
THOMAS, WA
[J]. JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1984, (02): : 155 - 164