SYNTHESIS OF THIENO[3,2-D]PYRIMIDINE-2,4-DIONES CYCLIC AND ACYCLIC NUCLEOSIDES AS POTENTIAL ANTI-HIV AGENTS

被引：18

作者：

JOURDAN, F

LADUREE, D

ROBBA, M

机构：

[1] Centre D'etudes Et de Recherche Sur Le Médicament de Normandie, U.F.R. Des Sciences Pharmaceutiques, Caen, 14032

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1994年 / 31卷 / 02期

关键词：

D O I：

10.1002/jhet.5570310208

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of cyclic and acyclic nucleosides was achieved by alkylation of 7-methyl or arylthieno[3,2-d]-pyrimidine-2,4-diones following the Vorbruggen and Niedballa's method [1]. After a possible deprotection, potential anti HIV agents were obtained.

引用

页码：305 / 312

页数：8

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