RELATIONSHIPS BETWEEN CSF DRUG CONCENTRATIONS, RECEPTOR-BINDING CHARACTERISTICS, AND PHARMACOKINETIC AND PHARMACODYNAMIC PROPERTIES OF SELECTED 1,4-SUBSTITUTED BENZODIAZEPINES

被引:21
作者
COLBURN, WA
JACK, ML
机构
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D O I
10.2165/00003088-198713030-00003
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:179 / 190
页数:12
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  • [1] AALTONEN L, 1980, ACTA PHARMACOL TOX, V46, P156
  • [2] BENZODIAZEPINES - CLINICAL-PHARMACOLOGY AND THERAPEUTIC USE
    BELLANTUONO, C
    REGGI, V
    TOGNONI, G
    GARATTINI, S
    [J]. DRUGS, 1980, 19 (03) : 195 - 219
  • [3] PHARMACOKINETICS OF ANTICONVULSANT DRUG CLONAZEPAM EVALUATED FROM SINGLE ORAL AND INTRAVENOUS DOSES AND BY REPEATED ORAL-ADMINISTRATION
    BERLIN, A
    DAHLSTROM, H
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1975, 9 (2-3) : 155 - 159
  • [4] COMPARATIVE PHARMACOKINETICS OF BENZODIAZEPINES IN DOG AND MAN
    BOXENBAUM, H
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1982, 10 (04): : 411 - 426
  • [5] PHARMACOKINETIC AND BIO-PHARMACEUTIC PROFILE OF CHLORDIAZEPOXIDE HCL IN HEALTHY SUBJECTS - SINGLE-DOSE STUDIES BY INTRAVENOUS, INTRAMUSCULAR, AND ORAL ROUTES
    BOXENBAUM, HG
    GEITNER, KA
    JACK, ML
    DIXON, WR
    SPIEGEL, HE
    SYMINGTON, J
    CHRISTIAN, R
    MOORE, JD
    WEISSMAN, L
    KAPLAN, SA
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1977, 5 (01): : 3 - 23
  • [6] PHARMACOLOGICAL CHARACTERIZATION OF BENZODIAZEPINE RECEPTORS IN BRAIN
    BRAESTRUP, C
    SQUIRES, RF
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (03) : 263 - 270
  • [7] BRAESTRUP C, 1980, TRENDS NEUROSCI, V3, P301
  • [8] BRAESTRUP C, 1980, ARZNEIMITTELFORSCH, V30-1, P852
  • [9] BRODIE BB, 1960, J PHARMACOL EXP THER, V130, P20
  • [10] SIMULTANEOUS PHARMACOKINETIC AND PHARMACODYNAMIC MODELING
    COLBURN, WA
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1981, 9 (03): : 367 - 388