PINACIDIL MONOHYDRATE - A NOVEL VASODILATOR - REVIEW OF PRECLINICAL PHARMACOLOGY AND MECHANISM OF ACTION

被引:16
作者
COHEN, ML
机构
关键词
D O I
10.1002/ddr.430090402
中图分类号
R914 [药物化学];
学科分类号
100701 ;
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页码:249 / 258
页数:10
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[1]   N''-CYANO-N-4-PYRIDYL-N'-1,2,2-TRIMETHYLPROPYLGUANIDINE, MONOHYDRATE (P 1134) - A NEW, POTENT VASODILATOR [J].
ARRIGONIMARTELLI, E ;
NIELSEN, CK ;
OLSEN, UB ;
PETERSEN, HJ .
EXPERIENTIA, 1980, 36 (04) :445-447
[2]   DIHYDROPYRIDINE RECEPTOR IN RAT-BRAIN LABELED WITH [H-3]-LABELED NIMODIPINE [J].
BELLEMANN, P ;
SCHADE, A ;
TOWART, R .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (08) :2356-2360
[3]   COMPARISON OF THE EFFECTS OF PINACIDIL AND ITS METABOLITE, PINACIDIL-N-OXIDE, IN ISOLATED SMOOTH AND CARDIAC-MUSCLE [J].
COHEN, ML ;
COLBERT, WE .
DRUG DEVELOPMENT RESEARCH, 1986, 7 (02) :111-124
[4]  
Dieperink H, 1983, J Hypertens, V1, P357, DOI 10.1097/00004872-198312000-00006
[5]   HYPOTENSIVE HYDRAZINOPHTHALAZINES AND RELATED COMPOUNDS [J].
DRUEY, J ;
MARXER, A .
JOURNAL OF MEDICINAL & PHARMACEUTICAL CHEMISTRY, 1959, 1 (01) :1-21
[6]   METABOLISM OF THE NEW ANTIHYPERTENSIVE AGENT PINACIDIL IN RAT, DOG AND MAN [J].
EILERTSEN, E ;
MAGNUSSEN, MP ;
PETERSEN, HJ ;
RASTRUPANDERSEN, N ;
SORENSEN, H ;
ARRIGONIMARTELLI, E .
XENOBIOTICA, 1982, 12 (03) :187-196
[7]   PHARMACOKINETICS AND DISTRIBUTION OF THE NEW ANTIHYPERTENSIVE AGENT PINACIDIL IN RAT, DOG AND MAN [J].
EILERTSEN, E ;
HART, JW ;
MAGNUSSEN, MP ;
SORENSEN, H ;
ARRIGONIMARTELLI, E .
XENOBIOTICA, 1982, 12 (03) :177-185
[8]  
FURCHGOTT RF, 1953, J PHARMACOL EXP THER, V108, P129
[9]   INHIBITION OF PLATELET-AGGREGATION AND THROMBOXANE PRODUCTION BY PINACIDIL [J].
GOODMAN, RP ;
LITTLE, DM ;
WRIGHT, JT .
PROSTAGLANDINS LEUKOTRIENES AND MEDICINE, 1985, 19 (02) :115-122
[10]  
GOODMAN RP, 1984, CLIN RES, V32, pA242