DOWN REGULATION OF SEROTONIN-S2 RECEPTOR-SITES IN RAT-BRAIN BY CHRONIC TREATMENT WITH THE SEROTONIN-S2 ANTAGONISTS - RITANSERIN AND SETOPERONE

被引:175
作者
LEYSEN, JE [1 ]
VANGOMPEL, P [1 ]
GOMMEREN, W [1 ]
WOESTENBORGHS, R [1 ]
JANSSEN, PAJ [1 ]
机构
[1] JANSSEN PHARMACEUT,DEPT CHIM,B-2340 BEERSE,BELGIUM
关键词
D O I
10.1007/BF00178504
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:434 / 444
页数:11
相关论文
共 34 条
[1]   DEVELOPMENT OF BETA-ADRENERGIC-RECEPTOR SUBSENSITIVITY BY ANTIDEPRESSANTS [J].
BANERJEE, SP ;
KUNG, LS ;
RIGGI, SJ ;
CHANDA, SK .
NATURE, 1977, 268 (5619) :455-456
[2]   ACUTE AND CHRONIC EFFECTS OF SEROTONIN (5HT) ANTAGONISTS ON SEROTONIN BINDING-SITES [J].
BLACKSHEAR, MA ;
FRIEDMAN, RL ;
SANDERSBUSH, E .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) :125-129
[3]  
BLACKSHEAR MA, 1982, J PHARMACOL EXP THER, V221, P303
[4]   EFFECT OF SEROTONIN ANTAGONISM IN SCHIZOPHRENIA - A PILOT-STUDY WITH SETOPERONE [J].
CEULEMANS, DLS ;
GELDERS, YG ;
HOPPENBROUWERS, MLJA ;
REYNTJENS, AJM ;
JANSSEN, PAJ .
PSYCHOPHARMACOLOGY, 1985, 85 (03) :329-332
[5]   BEHAVIORAL AND 5-HT ANTAGONIST EFFECTS OF RITANSERIN - A PURE AND SELECTIVE ANTAGONIST OF LSD DISCRIMINATION IN RAT [J].
COLPAERT, FC ;
MEERT, TF ;
NIEMEGEERS, CJE ;
JANSSEN, PAJ .
PSYCHOPHARMACOLOGY, 1985, 86 (1-2) :45-54
[6]  
Creese I, 1980, Adv Biochem Psychopharmacol, V24, P89
[7]   RAPID DOWN-REGULATION OF SEROTONIN2 RECEPTOR-BINDING DURING COMBINED ADMINISTRATION OF TRICYCLIC ANTI-DEPRESSANT DRUGS AND ALPHA-2-ANTAGONISTS [J].
CREWS, FT ;
SCOTT, JA ;
SHORSTEIN, NH .
NEUROPHARMACOLOGY, 1983, 22 (10) :1203-1209
[8]  
DECOURCELLES DD, 1985, J BIOL CHEM, V260, P7603
[9]   NICOTINIC ACETYLCHOLINE-RECEPTORS - AN OVERVIEW [J].
DOLLY, JO ;
BARNARD, EA .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (06) :841-858
[10]   DIFFERENT EFFECTS OF SEROTONIN ANTAGONISTS ON H-3 MIANSERIN AND H-3 KETANSERIN RECOGNITION SITES [J].
GANDOLFI, O ;
BARBACCIA, ML ;
COSTA, E .
LIFE SCIENCES, 1985, 36 (08) :713-721