AFFINITY OF CEPHALOSPORINS FOR BETA-LACTAMASES AS A FACTOR IN ANTIBACTERIAL EFFICACY

被引:89
作者
PHELPS, DJ [1 ]
CARLTON, DD [1 ]
FARRELL, CA [1 ]
KESSLER, RE [1 ]
机构
[1] BRISTOL MYERS CO LABS,DIV RES & DEV,DEPT MICROBIOL RES,SYRACUSE,NY 13221
关键词
D O I
10.1128/AAC.29.5.845
中图分类号
Q93 [微生物学];
学科分类号
071005 ; 100705 ;
摘要
引用
收藏
页码:845 / 848
页数:4
相关论文
共 15 条
[1]   INFLUENCE OF SPONTANEOUS AND INDUCIBLE BETA-LACTAMASE PRODUCTION ON THE ANTIMICROBIAL ACTIVITY OF RECENTLY DEVELOPED BETA-LACTAM COMPOUNDS [J].
CULLMANN, W ;
OPFERKUCH, W ;
STIEGLITZ, M ;
DICK, W .
CHEMOTHERAPY, 1984, 30 (03) :175-181
[2]   RELATION BETWEEN BETA-LACTAMASE PRODUCTION AND ANTI-MICROBIAL ACTIVITY - COMPARISON OF THE NEW COMPOUND HR-810 WITH CEFOTAXIME [J].
CULLMANN, W ;
OPFERKUCH, W ;
STIEGLITZ, M .
EUROPEAN JOURNAL OF CLINICAL MICROBIOLOGY & INFECTIOUS DISEASES, 1983, 2 (04) :350-352
[3]   THE DETERMINATION OF ENZYME INHIBITOR CONSTANTS [J].
DIXON, M .
BIOCHEMICAL JOURNAL, 1953, 55 (01) :170-171
[4]   A MODEL SYSTEM TO DEMONSTRATE THAT BETA-LACTAMASE ASSOCIATED ANTIBIOTIC TRAPPING COULD BE A POTENTIAL MEANS OF RESISTANCE [J].
GUTMANN, L ;
WILLIAMSON, R .
JOURNAL OF INFECTIOUS DISEASES, 1983, 148 (02) :316-321
[5]   COMPARISON OF A NEW CEPHALOSPORIN, BMY 28142, WITH OTHER BROAD-SPECTRUM BETA-LACTAM ANTIBIOTICS [J].
KESSLER, RE ;
BIES, M ;
BUCK, RE ;
CHISHOLM, DR ;
PURSIANO, TA ;
TSAI, YH ;
MISIEK, M ;
PRICE, KE ;
LEITNER, F .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1985, 27 (02) :207-216
[6]   NOVEL METHOD FOR DETECTION OF BETA-LACTAMASES BY USING A CHROMOGENIC CEPHALOSPORIN SUBSTRATE [J].
OCALLAGHAN, CH ;
SHINGLER, AH ;
KIRBY, SM ;
MORRIS, A .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1972, 1 (04) :283-+
[7]  
Richmond M H, 1973, Adv Microb Physiol, V9, P31, DOI 10.1016/S0065-2911(08)60376-8
[9]   CHROMOSOMAL BETA-LACTAMASES OF ENTEROBACTER-CLOACAE ARE RESPONSIBLE FOR RESISTANCE TO 3RD-GENERATION CEPHALOSPORINS [J].
SEEBERG, AH ;
TOLXDORFFNEUTZLING, RM ;
WIEDEMANN, B .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1983, 23 (06) :918-925
[10]   CEFOXITIN RESISTANCE BY A CHROMOSOMAL CEPHALOSPORINASE IN ESCHERICHIA-COLI [J].
TAKAHASHI, I ;
SAWAI, T ;
ANDO, T ;
YAMAGISHI, S .
JOURNAL OF ANTIBIOTICS, 1980, 33 (09) :1037-1042