SYNTHESIS OF A NOVEL CLASS OF HETEROAROMATIC AMINO-ACIDS AND THEIR USE IN THE PREPARATION OF ANALOGS OF LUTEINIZING-HORMONE-RELEASING HORMONE

被引：36

作者：

NESTOR, JJ ^{[1
]}

HORNER, BL ^{[1
]}

HO, TL ^{[1
]}

JONES, GH ^{[1
]}

MCRAE, GI ^{[1
]}

VICKERY, BH ^{[1
]}

机构：

[1] SYNTEX RES CORP,INST BIOL SCI,PALO ALTO,CA 94304

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1984年 / 27卷 / 03期

关键词：

D O I：

10.1021/jm00369a016

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：320 / 325

页数：6

共 36 条

[1]

ALBERT A, 1968, HETEROCYCLIC CHEM, P441

[2]

BERGMANN M, 1975, CHEM BER, V66, P1298

[3] OXIDATIVE REACTIONS OF HYDRAZINES .4. ELIMINATION OF NITROGEN FROM 1,1-DISUBSTITUTED-2-ARENESULFONHYDRAZIDES [J].

CARPINO, LA .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1957, 79 (16) :4427-4431

[4]

CORBIN A, 1975, ENDOCR RES COMMUN, V2, P1

[5] ANALOGS OF LUTEINIZING HORMONE-RELEASING HORMONE WITH INCREASED BIOLOGICAL-ACTIVITY PRODUCED BY D-AMINO-ACID SUBSTITUTIONS IN POSITION 6 [J].

COY, DH ;

VILCHEZMARTINEZ, JA ;

COY, EJ ;

SCHALLY, AV .

JOURNAL OF MEDICINAL CHEMISTRY, 1976, 19 (03) :423-425

[6] PEPTIDE ANTAGONISTS OF LH-RH - LARGE INCREASES IN ANTI-OVULATORY ACTIVITIES PRODUCED BY BASIC D-AMINO ACIDS IN THE 6 POSITION [J].

COY, DH ;

HORVATH, A ;

NEKOLA, MV ;

COY, EJ ;

ERCHEGYI, J ;

SCHALLY, AV .

ENDOCRINOLOGY, 1982, 110 (04) :1445-1447

[7] The titration constants of anserine, carnosine and some related compounds [J].

Deutsch, A ;

Eggleton, P .

BIOCHEMICAL JOURNAL, 1938, 32 :209-211

[8] UNUSUALLY STRONG LIPOPHILICITY OF FAT OR SUPER AMINO-ACIDS, INCLUDING A NEW REFERENCE VALUE FOR GLYCINE [J].

FAUCHERE, JL ;

DO, KQ ;

JOW, PYC ;

HANSCH, C .

EXPERIENTIA, 1980, 36 (10) :1203-1204

[9] USE OF NIM TERT BUTYLOXYCARBONYL IN SYNTHESIS OF POLY-L-HISTIDINE [J].

FRIDKIN, M ;

GOREN, HJ .

CANADIAN JOURNAL OF CHEMISTRY, 1971, 49 (09) :1578-&

[10] The solid-phase synthesis of ile(5)-angiotensin II to demonstrate the use of N-im-Tosyl-histidine [J].

Fujii, Toshiyuki ;

Sakakibara, Shurnpei .

BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, 1970, 43 (12) :3954A-3956

← 1 2 3 4 →