SELECTIVE ACTIVATION OF THE CONVERTING ENZYME-INHIBITOR MK 421 AND COMPARISON OF ITS ACTIVE DIACID FORM WITH CAPTOPRIL IN DIFFERENT TISSUES OF THE RAT

被引:81
作者
UNGER, T [1 ]
SCHULL, B [1 ]
RASCHER, W [1 ]
LANG, RE [1 ]
GANTEN, D [1 ]
机构
[1] UNIV HEIDELBERG,GERMAN INST HIGH BLOOD PRESSURE RES,D-6900 HEIDELBERG 1,FED REP GER
关键词
D O I
10.1016/0006-2952(82)90081-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3063 / 3070
页数:8
相关论文
共 15 条
[1]   EFFECT OF A NEW ANGIOTENSIN CONVERTING ENZYME-INHIBITOR MK 421 AND ITS LYSINE ANALOG ON THE COMPONENTS OF THE RENIN SYSTEM IN HEALTHY-SUBJECTS [J].
BRUNNER, DB ;
DESPONDS, G ;
BIOLLAZ, J ;
KELLER, I ;
FERBER, F ;
GAVRAS, H ;
BRUNNER, HR ;
SCHELLING, JL .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 11 (05) :461-467
[2]   FLUORIMETRIC DETERMINATION OF DIPEPTIDYL CARBOXYPEPTIDASE (ANGIOTENSIN-I-CONVERTING ENZYME) [J].
DEPIERRE, D ;
ROTH, M .
ENZYME, 1975, 19 (02) :65-70
[3]   ISO-RENIN OF EXTRARENAL ORIGIN - TISSUE ANGIOTENSINOGENASE SYSTEMS [J].
GANTEN, D ;
SCHELLING, P ;
VECSEI, P ;
GANTEN, U .
AMERICAN JOURNAL OF MEDICINE, 1976, 60 (06) :760-772
[4]  
GROSS DM, 1981, J PHARMACOL EXP THER, V216, P552
[5]   BLOOD-PRESSURE RESPONSES OF CONSCIOUS NORMOTENSIVE AND SPONTANEOUSLY HYPERTENSIVE RATS TO INTRACEREBROVENTRICULAR AND PERIPHERAL ADMINISTRATION OF CAPTOPRIL [J].
HUTCHINSON, JS ;
MENDELSOHN, FAO ;
DOYLE, AE .
HYPERTENSION, 1980, 2 (04) :546-550
[6]   EFFECT OF THE TIME INTERVAL BETWEEN BLOOD-SAMPLING AND ASSAY ON SERUM ANGIOTENSIN I-CONVERTING ENZYME-ACTIVITY FROM CAPTOPRIL-TREATED RATS [J].
LAI, FM ;
TANIKELLA, T ;
HERZLINGER, H ;
CERVONI, P .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 67 (01) :97-99
[7]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265
[8]   MECHANISM OF ANGIOTENSIN-I CONVERTING ENZYME-INHIBITION BY SQ20,881 (LESS-THAN GLU-TRP-PRO-ARG-PRO-GLN-ILE-PRO-PRO) INVIVO - FURTHER EVIDENCE FOR EXTRA-PULMONARY CONVERSION [J].
OPARIL, S ;
KOERNER, T ;
ODONOGHUE, JK .
HYPERTENSION, 1979, 1 (01) :13-22
[9]  
PATCHETT AA, 1980, NATURE, V288, P280, DOI 10.1038/288280a0
[10]   CONVERTING-ENZYME IN THE CHOROID-PLEXUS, BRAIN, AND KIDNEY - IMMUNO-CYTOCHEMICAL AND BIOCHEMICAL-STUDIES IN RATS [J].
RIX, E ;
GANTEN, D ;
SCHULL, B ;
UNGER, T ;
TAUGNER, R .
NEUROSCIENCE LETTERS, 1981, 22 (02) :125-130