BOP AS A REAGENT FOR MILD AND EFFICIENT PREPARATION OF ESTERS

被引：54

作者：

KIM, MH ^{[1
]}

PATEL, DV ^{[1
]}

机构：

[1] AFFYMAX RES INST,SANTA CLARA,CA 95051

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 31期

关键词：

D O I：

10.1016/S0040-4039(00)77257-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple procedure for preparation of esters under mild conditions employing the BOP reagent is reported. Acid and base labile protecting groups commonly used with amino acids e.g. t-butyl, Fmoc etc., are well tolerated under these conditions. The mechanism and scope of this reaction are briefly discussed.

引用

页码：5603 / 5606

页数：4

共 11 条

[1]

BODANSZKY M, 1981, SYNTHESIS-STUTTGART, P333

[2]

Bodanszky M., 1976, PEPTIDE SYNTHESIS

[3]

CAMPBELL DK, UNPUB

[4]

CASTRO B, 1975, TETRAHEDRON LETT, V14, P1219