A PROPOSAL FOR THE CLASSIFICATION OF SIGMA BINDING-SITES

被引:786
作者
QUIRION, R [1 ]
BOWEN, WD [1 ]
ITZHAK, Y [1 ]
JUNIEN, JL [1 ]
MUSACCHIO, JM [1 ]
ROTHMAN, RB [1 ]
SU, TP [1 ]
TAM, SW [1 ]
TAYLOR, DP [1 ]
机构
[1] MCGILL UNIV,DEPT PSYCHIAT,VERDUN H4H 1R3,QUEBEC,CANADA
关键词
D O I
10.1016/0165-6147(92)90030-A
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:85 / 86
页数:2
相关论文
共 41 条
[1]   EVIDENCE FOR A MULTI-SITE MODEL OF THE RAT-BRAIN SIGMA-RECEPTOR [J].
BOWEN, WD ;
HELLEWELL, SB ;
MCGARRY, KA .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1989, 163 (2-3) :309-318
[2]   METABOLITES OF HALOPERIDOL DISPLAY PREFERENTIAL ACTIVITY AT SIGMA-RECEPTORS COMPARED TO DOPAMINE D-2 RECEPTORS [J].
BOWEN, WD ;
MOSES, EL ;
TOLENTINO, PJ ;
WALKER, JM .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1990, 177 (03) :111-118
[3]  
BOWEN WD, IN PRESS MULTIPLE SI
[4]  
CAMPBELL BG, 1989, J NEUROSCI, V9, P3380
[6]   AUTORADIOGRAPHIC DISTRIBUTION OF NONDOPAMINERGIC BINDING-SITES LABELED [H-3] HALOPERIDOL IN RAT-BRAIN [J].
CONTRERAS, PC ;
QUIRION, R ;
GEHLERT, DR ;
CONTRERAS, ML ;
ODONOHUE, TL .
NEUROSCIENCE LETTERS, 1987, 75 (02) :133-140
[7]  
CRAVISO GL, 1983, MOL PHARMACOL, V23, P619
[8]  
CRAVISO GL, 1983, MOL PHARMACOL, V23, P629
[9]   SYNTHESIS AND EVALUATION OF OPTICALLY PURE [H-3] (+)-PENTAZOCINE, A HIGHLY POTENT AND SELECTIVE RADIOLIGAND FOR SIGMA-RECEPTORS [J].
DECOSTA, BR ;
BOWEN, WD ;
HELLEWELL, SB ;
WALKER, JM ;
THURKAUF, A ;
JACOBSON, AE ;
RICE, KC .
FEBS LETTERS, 1989, 251 (1-2) :53-58
[10]  
DIPAOLO L, 1991, SOC NEUR ABSTR, V17, P814