LIGAND-BINDING TO TRANSIENTLY ACCESSIBLE SITES - MECHANISMS FOR VARYING APPARENT BINDING RATES

被引:37
作者
STARMER, CF [1 ]
PACKER, DL [1 ]
GRANT, AO [1 ]
机构
[1] DUKE UNIV,MED CTR,DEPT COMP SCI,DURHAM,NC 27710
关键词
D O I
10.1016/S0022-5193(87)80120-0
中图分类号
Q [生物科学];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:335 / 341
页数:7
相关论文
共 10 条
[2]   NITRENDIPINE BLOCK OF CARDIAC CALCIUM CHANNELS - HIGH-AFFINITY BINDING TO THE INACTIVATED STATE [J].
BEAN, BP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (20) :6388-6392
[3]   FAST SODIUM CURRENT IN CARDIAC-MUSCLE - A QUANTITATIVE DESCRIPTION [J].
EBIHARA, L ;
JOHNSON, EA .
BIOPHYSICAL JOURNAL, 1980, 32 (02) :779-790
[5]   A QUANTITATIVE DESCRIPTION OF MEMBRANE CURRENT AND ITS APPLICATION TO CONDUCTION AND EXCITATION IN NERVE [J].
HODGKIN, AL ;
HUXLEY, AF .
JOURNAL OF PHYSIOLOGY-LONDON, 1952, 117 (04) :500-544
[6]   1,4-DIHYDROPYRIDINES AS TOOLS IN THE STUDY OF CA-2+ CHANNELS [J].
REUTER, H ;
PORZIG, H ;
KOKUBUN, S ;
PRODHOM, B .
TRENDS IN NEUROSCIENCES, 1985, 8 (09) :396-400
[7]  
STARMER CF, 1985, MOL PHARMACOL, V28, P348
[9]   A QUANTITATIVE DESCRIPTION OF QX222-BLOCKADE OF SODIUM-CHANNELS IN SQUID AXONS [J].
STARMER, CF ;
YEH, JZ ;
TANGUY, J .
BIOPHYSICAL JOURNAL, 1986, 49 (04) :913-920
[10]   NA CHANNEL ACTIVATION GATE MODULATES SLOW RECOVERY FROM USE-DEPENDENT BLOCK BY LOCAL-ANESTHETICS IN SQUID GIANT-AXONS [J].
YEH, JZ ;
TANGUY, J .
BIOPHYSICAL JOURNAL, 1985, 47 (05) :685-694