THE NOVEL ANTICONVULSANT MK-801 BINDS TO THE ACTIVATED STATE OF THE N-METHYL-D-ASPARTATE RECEPTOR IN RAT-BRAIN

被引:495
作者
FOSTER, AC
WONG, EHF
机构
关键词
D O I
10.1111/j.1476-5381.1987.tb10295.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:403 / 409
页数:7
相关论文
共 26 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]   ACETYLCHOLINE-RECEPTOR - AN ALLOSTERIC PROTEIN [J].
CHANGEUX, JP ;
DEVILLERSTHIERY, A ;
CHEMOUILLI, P .
SCIENCE, 1984, 225 (4668) :1335-1345
[3]   ANTICONVULSANT ACTIVITY OF (+)-5-METHYL-10, 11-DIHYDRO-5H-DIBENZO[A,D]CYCLOHEPTEN-5, 10-IMINE (MK-801), A SUBSTANCE WITH POTENT ANTICONVULSANT, CENTRAL SYMPATHOMIMETIC, AND APPARENT ANXIOLYTIC PROPERTIES [J].
CLINESCHMIDT, BV ;
MARTIN, GE ;
BUNTING, PR .
DRUG DEVELOPMENT RESEARCH, 1982, 2 (02) :123-134
[4]   [PHENCYCLIDINE-H-3 - A PROBE FOR THE IONIC CHANNEL OF THE NICOTINIC RECEPTOR [J].
ELDEFRAWI, ME ;
ELDEFRAWI, AT ;
ARONSTAM, RS ;
MALEQUE, MA ;
WARNICK, JE ;
ALBUQUERQUE, EX .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (12) :7458-7462
[5]   ACTIVATION, INACTIVATION, AND DESENSITIZATION OF ACETYLCHOLINE-RECEPTOR CHANNEL COMPLEX DETECTED BY BINDING OF PERHYDROHISTRIONICOTOXIN [J].
ELDEFRAWI, ME ;
ARONSTAM, RS ;
BAKRY, NM ;
ELDEFRAWI, AT ;
ALBUQUERQUE, EX .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2309-2313
[6]   ANTAGONISM OF EXCITATORY AMINO ACID-INDUCED RESPONSES AND OF SYNAPTIC EXCITATION IN THE ISOLATED SPINAL-CORD OF THE FROG [J].
EVANS, RH ;
FRANCIS, AA ;
HUNT, K ;
OAKES, DJ ;
WATKINS, JC .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 67 (04) :591-603
[7]   THE EFFECTS OF A SERIES OF OMEGA-PHOSPHONIC ALPHA-CARBOXYLIC AMINO-ACIDS ON ELECTRICALLY EVOKED AND EXCITANT AMINO ACID-INDUCED RESPONSES IN ISOLATED SPINAL-CORD PREPARATIONS [J].
EVANS, RH ;
FRANCIS, AA ;
JONES, AW ;
SMITH, DAS ;
WATKINS, JC .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (01) :65-75
[8]   SELECTIVE ASSOCIATION OF N-METHYL ASPARTATE AND QUISQUALATE TYPES OF L-GLUTAMATE RECEPTOR WITH BRAIN POSTSYNAPTIC DENSITIES [J].
FAGG, GE ;
MATUS, A .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (21) :6876-6880
[9]  
FOSTER A C, 1986, British Journal of Pharmacology, V89, p869P
[10]   ACIDIC AMINO-ACID BINDING-SITES IN MAMMALIAN NEURONAL MEMBRANES - THEIR CHARACTERISTICS AND RELATIONSHIP TO SYNAPTIC RECEPTORS [J].
FOSTER, AC ;
FAGG, GE .
BRAIN RESEARCH REVIEWS, 1984, 7 (02) :103-164