DESIGN, SYNTHESIS AND BIOASSAYS OF ANTAGONISTS OF LHRH WHICH HAVE HIGH ANTIOVULATORY ACTIVITY AND RELEASE NEGLIGIBLE HISTAMINE

被引：63

作者：

LJUNGQVIST, A

FENG, DM

TANG, PFL

KUBOTA, M

OKAMOTO, T

ZHANG, YW

BOWERS, CY

FOLKERS, K

机构：

[1] TULANE UNIV,SCH MED,ENDOCRINE UNIT,NEW ORLEANS,LA 70112

[2] NIDR,BETHESDA,MD 20892

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1987年 / 148卷 / 02期

关键词：

D O I：

10.1016/0006-291X(87)90953-3

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：849 / 856

页数：8

共 11 条

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[2] FOLKERS K, 1984, BIOCHEM BIOPH RES CO, V123, P1221, DOI 10.1016/S0006-291X(84)80263-6
[3] INCREASED POTENCY OF ANTAGONISTS OF THE LUTEINIZING-HORMONE-RELEASING HORMONE WHICH HAVE D-3-PAL IN POSITION-6
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[4] EFFECT OF REDUCTIVE ALKYLATION OF D-LYSINE IN POSITION 6 ON THE HISTAMINE-RELEASING ACTIVITY OF LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONISTS
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[5] HOOK WA, 1985, FED PROC, V44, P1323
[6] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF LH-RH ANTAGONISTS MODIFIED IN POSITION-1
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COY, EJ
SCHALLY, AV
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[J]. PEPTIDES, 1982, 3 (06) : 969 - 971
[7] PEPTIDE HORMONES .109. INHIBITORY ANALOGS OF LUTEINIZING-HORMONE-RELEASING HORMONE HAVING D-AROMATIC RESIDUES IN POSITIONS 2 AND 6 AND VARIATION IN POSITION 3
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[8] GONADOTROPIN-RELEASING-HORMONE ANALOG DESIGN - STRUCTURE-FUNCTION STUDIES TOWARD THE DEVELOPMENT OF AGONISTS AND ANTAGONISTS - RATIONALE AND PERSPECTIVE
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RIVIER, JE
[J]. ENDOCRINE REVIEWS, 1986, 7 (01) : 44 - 66
[9] KARTEN MJ, 1987, LHRH ITS ANALOGS CON, V2, P179
[10] LUTEINIZING-HORMONE-RELEASING HORMONE ANTAGONISTS CONTAINING VERY HYDROPHOBIC AMINO-ACIDS
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (09) : 1170 - 1174

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