PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA .15. (3S,4S)-(+)-TRANS-3-METHYLFENTANYL ISOTHIOCYANATE, A POTENT SITE-DIRECTED ACYLATING AGENT FOR THE DELTA-OPIOID RECEPTORS INVITRO

被引:28
作者
KIM, CH
ROTHMAN, RB
JACOBSON, AE
MATTSON, MV
BYKOV, V
STREATY, RA
KLEE, WA
GEORGE, C
LONG, JB
RICE, KC
机构
[1] NIDDK, MED CHEM LAB, BETHESDA, MD 20892 USA
[2] NIMH, MOLEC BIOL LAB, BETHESDA, MD 20892 USA
[3] NIMH, CLIN SCI LAB, BETHESDA, MD 20892 USA
[4] USN, RES LAB, STRUCT MATTER LAB, WASHINGTON, DC 20375 USA
[5] WALTER REED ARMY INST RES, NEUROPHARMACOL BRANCH, WASHINGTON, DC 20307 USA
关键词
D O I
10.1021/jm00126a040
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1392 / 1398
页数:7
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