THE EFFECTS OF ENZYME-INDUCTION AND ENZYME-INHIBITION ON LABETALOL PHARMACOKINETICS

被引:29
作者
DANESHMEND, TK [1 ]
ROBERTS, CJC [1 ]
机构
[1] UNIV BRISTOL,BRISTOL ROYAL INFIRM,DEPT MED,BRISTOL BS2 8HW,AVON,ENGLAND
关键词
D O I
10.1111/j.1365-2125.1984.tb02481.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:393 / 400
页数:8
相关论文
共 21 条
  • [1] INCREASED CLEARANCE OF ANTIPYRINE AND D-PROPRANOLOL AFTER PHENOBARBITAL TREATMENT IN MONKEY - RELATIVE CONTRIBUTIONS OF ENZYME-INDUCTION AND INCREASED HEPATIC BLOOD-FLOW
    BRANCH, RA
    SHAND, DG
    WILKINSON, GR
    NIES, AS
    [J]. JOURNAL OF CLINICAL INVESTIGATION, 1974, 53 (04) : 1101 - 1107
  • [2] EFFECTS OF CHRONIC ORAL CIMETIDINE ON APPARENT LIVER BLOOD-FLOW AND HEPATIC MICROSOMAL-ENZYME ACTIVITY IN MAN
    DANESHMEND, TK
    ENE, MD
    PARKER, G
    ROBERTS, CJC
    [J]. GUT, 1984, 25 (02) : 125 - 128
  • [3] DESMOND PV, 1981, GASTROENTEROLOGY, V80, P1330
  • [4] REDUCTION OF LIVER BLOOD-FLOW AND PROPRANOLOL METABOLISM BY CIMETIDINE
    FEELY, J
    WILKINSON, GR
    WOOD, AJJ
    [J]. NEW ENGLAND JOURNAL OF MEDICINE, 1981, 304 (12) : 692 - 695
  • [5] FINE A, 1981, CAN MED ASSOC J, V124, P1434
  • [6] INFLUENCE OF CIMETIDINE ON PHARMACOKINETICS OF PROPRANOLOL
    HEAGERTY, AM
    DONOVAN, MA
    CASTLEDEN, CM
    POHL, JF
    PATEL, L
    HEDGES, A
    [J]. BRITISH MEDICAL JOURNAL, 1981, 282 (6280) : 1917 - 1919
  • [7] DECREASED 1ST-PASS METABOLISM OF LABETALOL IN CHRONIC LIVER-DISEASE
    HOMEIDA, M
    JACKSON, L
    ROBERTS, CJC
    [J]. BRITISH MEDICAL JOURNAL, 1978, 2 (6144) : 1048 - 1050
  • [8] FEATURES OF HEPATIC ENZYME-INDUCTION WITH GLUTETHIMIDE IN MAN
    JACKSON, L
    HOMEIDA, M
    ROBERTS, CJC
    [J]. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1978, 6 (06) : 525 - 528
  • [9] INFLUENCE OF CIMETIDINE ON THE PHARMACOKINETICS OF DESMETHYLDIAZEPAM AND OXAZEPAM
    KLOTZ, U
    REIMANN, I
    [J]. EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 18 (06) : 517 - 520
  • [10] MARTIN LE, 1976, BRIT J CLIN PHARMACO, V3, pS695