THE GAMMA-AMINOBUTYRATE BENZODIAZEPINE RECEPTOR FROM PIG BRAIN - ENHANCEMENT OF GAMMA-AMINOBUTYRATE-RECEPTOR BINDING BY THE ANESTHETIC PROPANIDID

被引:20
作者
KIRKNESS, EF [1 ]
TURNER, AJ [1 ]
机构
[1] UNIV LEEDS,DEPT BIOCHEM,LEEDS LS2 9JT,W YORKSHIRE,ENGLAND
关键词
D O I
10.1042/bj2330259
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:259 / 264
页数:6
相关论文
共 35 条
[1]   STIMULATION OF GABA RECEPTOR-BINDING BY BARBITURATES [J].
ASANO, T ;
OGASAWARA, N .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 77 (04) :355-357
[2]   CHLORIDE-DEPENDENT STIMULATION OF GABA AND BENZODIAZEPINE RECEPTOR-BINDING BY PENTOBARBITAL [J].
ASANO, T ;
OGASAWARA, N .
BRAIN RESEARCH, 1981, 225 (01) :212-216
[3]   ETOMIDATE STEREOSPECIFICALLY STIMULATES FOREBRAIN, BUT NOT CEREBELLAR, DIAZEPAM-H-3 BINDING [J].
ASHTON, D ;
GEERTS, R ;
WATERKEYN, C ;
LEYSEN, JE .
LIFE SCIENCES, 1981, 29 (25) :2631-2636
[4]   MUSCIMOL BINDING IN RAT-BRAIN - ASSOCIATION WITH SYNAPTIC GABA RECEPTORS [J].
BEAUMONT, K ;
CHILTON, WS ;
YAMAMURA, HI ;
ENNA, SJ .
BRAIN RESEARCH, 1978, 148 (01) :153-162
[5]   DIFFERENTIAL EFFECTS OF TRITON X-100 ON BENZODIAZEPINE AND GABA BINDING IN A FROZEN-THAWED SYNAPTOSOMAL FRACTION OF RAT-BRAIN [J].
CHIU, TH ;
ROSENBERG, HC .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 58 (03) :335-338
[6]   PROPANIDID [J].
CONWAY, CM ;
ELLIS, DB .
BRITISH JOURNAL OF ANAESTHESIA, 1970, 42 (03) :249-&
[7]   EXPERIMENTAL STUDIES OF BREAKDOWN OF EPONTOL - DETERMINATION OF PROPANIDID IN HUMAN SERUM [J].
DOENICKE, A ;
KRUMEY, I ;
KUGLER, J ;
KLEMPA, J .
BRITISH JOURNAL OF ANAESTHESIA, 1968, 40 (06) :415-&
[8]  
ENNA SJ, 1977, MOL PHARMACOL, V13, P442
[9]   GABA-MIMETIC ACTION OF ETOMIDATE [J].
EVANS, RH ;
HILL, RG .
EXPERIENTIA, 1978, 34 (10) :1325-1327
[10]   SOLUBILIZATION OF HISTAMINE H-1, GABA AND BENZODIAZEPINE RECEPTORS [J].
GAVISH, M ;
CHANG, RSL ;
SNYDER, SH .
LIFE SCIENCES, 1979, 25 (09) :783-789