EFFECTS OF FORMULATION ON THE PHARMACOKINETICS OF ORALLY-ADMINISTERED PINACIDIL IN HUMANS

被引:6
作者
MCBURNEY, A [1 ]
FARROW, PR [1 ]
WARD, JW [1 ]
机构
[1] PFIZER LTD,CENT RES,RES DEPT,SANDWICH CT13 9NJ,KENT,ENGLAND
关键词
D O I
10.1002/jps.2600761220
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:940 / 941
页数:2
相关论文
共 10 条
[1]   N''-CYANO-N-4-PYRIDYL-N'-1,2,2-TRIMETHYLPROPYLGUANIDINE, MONOHYDRATE (P 1134) - A NEW, POTENT VASODILATOR [J].
ARRIGONIMARTELLI, E ;
NIELSEN, CK ;
OLSEN, UB ;
PETERSEN, HJ .
EXPERIENTIA, 1980, 36 (04) :445-447
[2]   PINACIDIL, A NEW VASODILATOR - PHARMACOKINETICS AND PHARMACODYNAMICS OF A NEW RETARDED RELEASE TABLET IN ESSENTIAL-HYPERTENSION [J].
CARLSEN, JE ;
KARDEL, T ;
JENSEN, HA ;
TANGO, M ;
TRAPJENSEN, J .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1983, 25 (04) :557-561
[3]  
CARLSEN JE, 1981, J CLIN PHYSL, V1, P357
[4]   THE EFFECTS OF LONG-ACTING PINACIDIL ON INTRA-ARTERIAL BLOOD-PRESSURE [J].
CARUANA, MP ;
ALKHAWAJA, I ;
ROYSTON, P ;
RAFTERY, EB .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1985, 20 (02) :140-143
[5]   METABOLISM OF THE NEW ANTIHYPERTENSIVE AGENT PINACIDIL IN RAT, DOG AND MAN [J].
EILERTSEN, E ;
MAGNUSSEN, MP ;
PETERSEN, HJ ;
RASTRUPANDERSEN, N ;
SORENSEN, H ;
ARRIGONIMARTELLI, E .
XENOBIOTICA, 1982, 12 (03) :187-196
[6]   N''-CYANO-N-4-PYRIDYL-N'-1,2,2-TRIMETHYL-PROPYLGUANIDINE, A NEW VASODILATING AGENT - ACUTE EFFECT ON BLOOD-PRESSURE AND PHARMACOKINETICS IN HYPERTENSIVE PATIENTS [J].
KARDEL, T ;
HILDEN, T ;
CARLSEN, J ;
TRAPJENSEN, J .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1981, 3 (05) :1002-1007
[7]  
MUIESAN G, 1983, CLIN PHARMACOL THER, V33, P229
[8]   PRELIMINARY EVALUATION OF PINACIDIL IN HYPERTENSION [J].
RAMSAY, LE ;
FREESTONE, S .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1983, 16 (03) :336-338
[9]   PHARMACOKINETICS AND HYPOTENSIVE EFFECT IN HEALTHY-VOLUNTEERS OF PINACIDIL, A NEW POTENT VASODILATOR [J].
WARD, JW ;
MCBURNEY, A ;
FARROW, PR ;
SHARP, P .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 26 (05) :603-608
[10]   PINACIDIL MONOTHERAPY FOR HYPERTENSION [J].
WARD, JW .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 18 (02) :223-225