CYANOPINDOLOL IS A HIGHLY POTENT AND SELECTIVE ANTAGONIST AT THE PRESYNAPTIC SEROTONIN AUTORECEPTOR IN THE RAT-BRAIN CORTEX

被引:42
作者
SCHLICKER, E [1 ]
GOTHERT, M [1 ]
HILLENBRAND, K [1 ]
机构
[1] UNIV ESSEN GESAMTHSCH,INST PHARMAKOL,HUFELANDSTR 55,D-4300 ESSEN 1,FED REP GER
关键词
D O I
10.1007/BF00500826
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:398 / 401
页数:4
相关论文
共 20 条
[1]   FURTHER EVIDENCE FOR NEGATIVE FEEDBACK-CONTROL OF SEROTONIN RELEASE IN THE CENTRAL NERVOUS-SYSTEM [J].
BAUMANN, PA ;
WALDMEIER, PC .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 317 (01) :36-43
[2]   EVIDENCE FOR COMMON PHARMACOLOGICAL PROPERTIES OF [H-3]5-HYDROXYTRYPTAMINE BINDING-SITES, PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE AUTORECEPTORS IN CNS AND INHIBITORY PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE RECEPTORS ON SYMPATHETIC-NERVES [J].
ENGEL, G ;
GOTHERT, M ;
MULLERSCHWEINITZER, E ;
SCHLICKER, E ;
SISTONEN, L ;
STADLER, PA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) :116-124
[3]  
ENGEL G, 1985, NAUNYNSCHMIEDEBERGS
[4]   NORADRENALINE INHIBITS DEPOLARIZATION-INDUCED SEROTONIN-H-3 RELEASE FROM SLICES OF RAT HIPPOCAMPUS [J].
FRANKHUYZEN, AL ;
MULDER, AH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1980, 63 (2-3) :179-182
[5]  
Furchgott RF, 1972, HDB EXPT PHARM, V3, P283
[6]   EXTRACELLULAR 5-HYDROXYTRYPTAMINE INHIBITS 5-HYDROXYTRYPTAMINE RELEASE FROM RAT-BRAIN CORTEX SLICES [J].
GOTHERT, M ;
WEINHEIMER, G .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 310 (01) :93-96
[8]  
GOTHERT M, 1985, VASCULAR NEUROEFFECT, P315
[9]  
HERY F, 1981, J PHYSIOLOGY PARIS, V77, P287
[10]   MODULATION OF NORADRENALINE RELEASE THROUGH ACTIVATION OF PRE-SYNAPTIC BETA-ADRENORECEPTORS [J].
MAJEWSKI, H .
JOURNAL OF AUTONOMIC PHARMACOLOGY, 1983, 3 (01) :47-60